SCHEMBL8974338

SCHEMBL8974338

NS(=O)(=O)c1ccc(C2=CCC=C2c2ccc(Cl)cc2)cn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 9/20 0.44
CA2 P00918 9/20 0.44
CA9 Q16790 7/20 0.44
CA12 O43570 5/20 0.44
CA4 P22748 5/20 0.44
CA7 P43166 4/20 0.44
CA5A P35218 3/20 0.44
CA13 Q8N1Q1 3/20 0.44
CA6 P23280 2/20 0.44
CA14 Q9ULX7 2/20 0.44
CA5B Q9Y2D0 2/20 0.39
PTGS2 P35354 9/20 0.38
PTGS1 P23219 5/20 0.38
MAOB P27338 2/20 0.37
MAOA P21397 1/20 0.37
CA3 P07451 1/20 0.37
IKBKB O14920 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8973795 0.87 CA1 (0.45) CA1CA2CA9CA12CA4
SCHEMBL8974334 0.85 CA1 (0.44) CA1CA2CA9CA12CA4
SCHEMBL8974603 0.85 FAAH (0.41) PTGS2PTGS1NPC1RAB9ARXFP1
SCHEMBL8973749 0.85 CA1 (0.44) CA1CA2CA9CA12CA4
SCHEMBL9115309 0.82 CA1 (0.41) CA1CA2CA9CA12CA4
SCHEMBL8974062 0.82 KIF11 (0.45) CA1CA2CA9CA12CA4
SCHEMBL8974661 0.82 CA1 (0.45) CA1CA2CA9CA12CA4
SCHEMBL9119047 0.80 CA1 (0.39) CA1CA2CA9CA12CA4
SCHEMBL9117244 0.80 CA1 (0.39) CA1CA2CA9CA12CA4
SCHEMBL8974750 0.78 CA2 (0.64) CA1CA2CA9CA12CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO claimed
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed