SCHEMBL8974448

SCHEMBL8974448

CS(=O)(=O)c1ccc(C2=CCC=C2c2ccc(C#N)cn2)cc1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.48
GPR119 Q8TDV5 1/20 0.45
ATR Q13535 1/20 0.41
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 2/20 0.38
HTT P42858 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CCR6 P51684 3/20 0.37
MLNR O43193 1/20 0.37
LRRK2 Q5S007 2/20 0.37
KDM1A O60341 1/20 0.37
KIT P10721 1/20 0.36
TNKS O95271 1/20 0.36
TNKS2 Q9H2K2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974590 0.93 PTGS2 (0.48) PTGS2GPR119ATRMLNRKDM1A
SCHEMBL8974324 0.88 CA2 (0.52) PTGS2CCR6MLNRKDM1A
SCHEMBL8974143 0.85 PTGS2 (0.63) PTGS2GPR119
SCHEMBL8974082 0.82 CA2 (0.52) PTGS2MLNRKDM1A
SCHEMBL9116993 0.82 PTGS2 (0.54) PTGS2GPR119ATRKDM4EALDH1A1
SCHEMBL8974359 0.82 PTGS2 (0.55) PTGS2GPR119
SCHEMBL8974116 0.81 PTGS2 (0.44) PTGS2GPR119
SCHEMBL8974412 0.81 PTGS2 (0.48) PTGS2GPR119
SCHEMBL9117705 0.80 PTGS2 (0.49) PTGS2GPR119ATRKDM4EALDH1A1
SCHEMBL8973819 0.79 PTGS2 (0.46) PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed