SCHEMBL9116993

SCHEMBL9116993

CS(=O)(=O)c1ccc(C2=CC3(C=C2c2ccc(C#N)cn2)CC3)cc1

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.54
PTGS1 P23219 2/20 0.54
GPR119 Q8TDV5 1/20 0.45
ATR Q13535 1/20 0.40
CCR6 P51684 4/20 0.38
LRRK2 Q5S007 5/20 0.37
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
HPGD P15428 2/20 0.36
HTT P42858 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9117705 0.95 PTGS2 (0.49) PTGS2PTGS1GPR119ATRCCR6
SCHEMBL9117672 0.93 PTGS2 (0.51) PTGS2PTGS1GPR119ATRCCR6
SCHEMBL9117491 0.89 PTGS2 (0.46) PTGS2PTGS1GPR119ATRCCR6
SCHEMBL9116434 0.89 PTGS2 (0.46) PTGS2PTGS1GPR119ATRCCR6
SCHEMBL9115957 0.88 CA2 (0.49) PTGS2PTGS1CCR6
SCHEMBL9118956 0.84 CA2 (0.47) PTGS2PTGS1CCR6
SCHEMBL9115333 0.84 CA2 (0.47) PTGS2PTGS1CCR6
SCHEMBL9117633 0.84 CA2 (0.49) PTGS2PTGS1ATRCCR6
SCHEMBL9117836 0.83 PTGS2 (0.59) PTGS2PTGS1GPR119
SCHEMBL8974448 0.82 PTGS2 (0.48) PTGS2GPR119ATRCCR6LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995030652-A1 SUBSTITUTED SPIRODIENES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed