SCHEMBL8974753

SCHEMBL8974753

NS(=O)(=O)c1ccc(C2=CC(CO)(CO)C=C2c2ccc(C(F)(F)F)cc2)cn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 6/20 0.40
MAP4K4 O95819 1/20 0.38
ALOX5AP P20292 5/20 0.38
FEN1 P39748 5/20 0.38
POLB P06746 1/20 0.37
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA4 P22748 1/20 0.36
CA6 P23280 1/20 0.36
CA5A P35218 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
CA13 Q8N1Q1 1/20 0.36
CA14 Q9ULX7 1/20 0.36
PPARD Q03181 1/20 0.36
PTGS2 P35354 3/20 0.36
PTGS1 P23219 2/20 0.36
COMT P21964 1/20 0.34
SLC22A12 Q96S37 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974461 0.89 KIF11 (0.41) KIF11MAP4K4ALOX5APFEN1POLB
SCHEMBL8974809 0.88 PTGS2 (0.40) MAP4K4ALOX5APFEN1POLBPPARD
SCHEMBL8973783 0.88 KIF11 (0.40) KIF11ALOX5APFEN1POLBCA12
SCHEMBL8974086 0.86 CA1 (0.42) MAP4K4CA12CA1CA2CA4
SCHEMBL8973844 0.86 KIF11 (0.40) KIF11MAP4K4ALOX5APFEN1POLB
SCHEMBL9131829 0.84 KIF11 (0.43) KIF11ALOX5APFEN1POLBCA12
SCHEMBL9117838 0.84 KIF11 (0.43) KIF11ALOX5APFEN1POLBCA12
SCHEMBL9118048 0.83 PTGS2 (0.42) KIF11ALOX5APFEN1POLBCA12
SCHEMBL8973750 0.82 KIF11 (0.62) KIF11CA12CA1CA2CA4
SCHEMBL8973763 0.81 POLB (0.41) KIF11POLBCA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed