SCHEMBL8974889

SCHEMBL8974889

NS(=O)(=O)c1ccc(C2=CCC=C2c2ccccc2)nc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 13/20 0.45
CA1 P00915 11/20 0.45
CA9 Q16790 10/20 0.45
CA12 O43570 8/20 0.45
CA5A P35218 3/20 0.42
CA5B Q9Y2D0 3/20 0.42
CA4 P22748 2/20 0.42
CA7 P43166 2/20 0.41
FLT1 P17948 1/20 0.41
FLT4 P35916 1/20 0.41
KDR P35968 1/20 0.41
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
PTGS2 P35354 5/20 0.39
IKBKB O14920 1/20 0.39
TDP1 Q9NUW8 1/20 0.38
CA3 P07451 1/20 0.38
CA6 P23280 1/20 0.38
PLA2G7 Q13093 1/20 0.38
CA13 Q8N1Q1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974157 0.86 CA2 (0.45) CA2CA1CA9CA5ACA5B
SCHEMBL8974882 0.86 CA2 (0.45) CA2CA1CA9CA12CA5A
SCHEMBL8974679 0.86 PTGS2 (0.47) CA2CA1CA9CA12CA5A
SCHEMBL8974156 0.86 PTGS2 (0.41) PTGS2PTGS1
SCHEMBL8974082 0.83 CA2 (0.52) CA2CA1CA9CA12CA4
SCHEMBL8974067 0.83 KIF11 (0.52) CA2CA1CA9CA12CA4
SCHEMBL18191710 0.81 CA1 (0.57) CA2CA1CA9CA12CA5A
SCHEMBL8974782 0.81 CA2 (0.68) CA2CA1CA9CA12CA5A
SCHEMBL8974823 0.81 PTGS2 (0.56) CA2CA1CA9CA12CA5A
SCHEMBL8973735 0.81 CA2 (0.45) CA2CA1CA9CA12CA5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed