SCHEMBL8974969

SCHEMBL8974969

O=C(O)c1cccc(N(S(=O)(=O)c2ccc3ccccc3c2)S(=O)(=O)c2ccc3ccccc3c2)c1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.53
ALDH1A1 P00352 2/20 0.50
LMNA P02545 1/20 0.50
KAT6A Q92794 2/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
SLC16A3 O15427 4/20 0.46
HTR2C P28335 1/20 0.46
HTR6 P50406 1/20 0.46
MCL1 Q07820 3/20 0.46
PTGES O14684 1/20 0.46
ALOX5 P09917 1/20 0.46
POLB P06746 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
MRGPRX4 Q96LA9 1/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
BCL2L1 Q07817 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8973992 0.85 ALDH1A1 (0.57) AKR1C3ALDH1A1LMNAMEN1KMT2A
SCHEMBL8973935 0.84 PLAU (0.58) ALDH1A1LMNAKAT6ANPC1RAB9A
SCHEMBL18392260 0.80 MCL1 (0.70) ALDH1A1LMNAMCL1MEN1KMT2A
SCHEMBL30076572 0.80 MCL1 (0.70) ALDH1A1LMNAMCL1MEN1KMT2A
SCHEMBL7186113 0.77 ALDH1A1 (0.47) AKR1C3ALDH1A1LMNAKAT6ANPC1
SCHEMBL7513281 0.76 HTR2C (0.47) ALDH1A1LMNAKAT6ANPC1RAB9A
SCHEMBL3872842 0.76 POLB (0.53) AKR1C3ALDH1A1LMNANPC1RAB9A
SCHEMBL5928513 0.75 AKR1C3 (0.47) AKR1C3ALDH1A1LMNASLC16A3PTGES
SCHEMBL7103484 0.74 MEN1 (0.52) ALDH1A1LMNAKAT6ANPC1RAB9A
SCHEMBL8974735 0.74 MCL1 (0.50) AKR1C3ALDH1A1LMNAKAT6ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996039132-A1 N,N-DISULFONYLATED AMINOBENZENE CARBOXYLIC ACIDS AND THE USE THEREOF AS THROMBIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 1996-12-12 WO disclosed
US-5559150-A ANTICOAGULANT, ANTITUMOR, ANTIINFLAMMATORY 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 1996-09-24 US disclosed
WO-1996002517-A1 SUBSTITUTED ARYLSULFONAMIDES, THEIR PREPARATION AND USE AS THROMBIN-INHIBITING MEDICAMENTS DR. KARL THOMAE GMBH (DE) 1996-02-01 WO disclosed