SCHEMBL7513281

SCHEMBL7513281

O=S(=O)(c1cc(Cl)cc(Cl)c1)N(c1cccc(N(S(=O)(=O)c2ccc3ccccc3c2)S(=O)(=O)c2ccc3ccccc3c2)c1)S(=O)(=O)c1cc(Cl)cc(Cl)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 4/20 0.47
HTR6 P50406 4/20 0.47
VCAM1 P19320 1/20 0.47
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
S1PR1 P21453 1/20 0.44
L3MBTL1 Q9Y468 3/20 0.43
POLB P06746 2/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.42
HTR2A P28223 3/20 0.42
DRD3 P35462 3/20 0.42
HTR1A P08908 2/20 0.42
HTR7 P34969 2/20 0.42
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
KAT6A Q92794 2/20 0.40
HTT P42858 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
CNR2 P34972 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7103481 0.86 HTR2C (0.41) HTR2CHTR6VCAM1NPC1RAB9A
SCHEMBL7103484 0.81 MEN1 (0.52) NPC1RAB9AL3MBTL1ALDH1A1LMNA
SCHEMBL7101292 0.79 PGR (0.46) ALDH1A1MEN1KMT2AHTTNPSR1
SCHEMBL8974969 0.76 AKR1C3 (0.53) HTR2CHTR6NPC1RAB9AL3MBTL1
SCHEMBL7098960 0.75 TP53 (0.50) POLBALDH1A1LMNANPSR1
SCHEMBL7517997 0.74 S1PR1 (0.44) VCAM1S1PR1ALDH1A1LMNAMEN1
SCHEMBL13602324 0.72 MEN1 (0.49) HTR2CHTR6VCAM1NPC1RAB9A
SCHEMBL8973935 0.72 PLAU (0.58) HTR2CHTR6NPC1RAB9APOLB
SCHEMBL13690005 0.71 NPC1 (0.48) HTR2CHTR6VCAM1NPC1RAB9A
SCHEMBL11507803 0.71 LMNA (0.57) HTR2CHTR6NPC1RAB9AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020127605-A1 Bisubstituted carbocyclic cyclophilin binding compounds and their use GUILFORD PHARMACEUTICALS, INC. 2002-09-12 US claimed
US-20020127605-A1 Bisubstituted carbocyclic cyclophilin binding compounds and their use GUILFORD PHARMACEUTICALS, INC. 2002-09-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020127605-A1 Bisubstituted carbocyclic cyclophilin binding compounds and their use PPIG, PIN1, PPIH HTR2C 1745/4885HTR6 3151/4885VCAM1 1999/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.