SCHEMBL8975003

SCHEMBL8975003

NCCC=Cc1ccc(F)cc1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 7/20 0.46
HSD11B1 P28845 1/20 0.42
GRIK1 P39086 1/20 0.41
GRIK2 Q13002 1/20 0.41
TAAR1 Q96RJ0 1/20 0.41
APP P05067 1/20 0.41
PTGS1 P23219 1/20 0.41
FBP1 P09467 1/20 0.39
LOXL2 Q9Y4K0 1/20 0.39
DRD2 P14416 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5728588 0.88 NFE2L2 (0.43) NFE2L2HSD11B1GRIK1GRIK2TAAR1
SCHEMBL10423140 0.82 NFE2L2 (0.50) NFE2L2HSD11B1GRIK1GRIK2APP
SCHEMBL17862090 0.81 NFE2L2 (0.59) NFE2L2HSD11B1APPPTGS1FBP1
SCHEMBL8325205 0.78 AHR (0.45) NFE2L2GRIK1GRIK2TAAR1PTGS1
SCHEMBL5682382 0.78 AHR (0.45) NFE2L2GRIK1GRIK2TAAR1PTGS1
SCHEMBL7423750 0.78 NFE2L2 (0.46) NFE2L2HSD11B1APPPTGS1FBP1
SCHEMBL9663338 0.78 NFE2L2 (0.46) NFE2L2HSD11B1APPPTGS1FBP1
SCHEMBL7097687 0.78 HSD11B1 (0.47) NFE2L2HSD11B1GRIK1GRIK2APP
SCHEMBL7097682 0.78 HSD11B1 (0.47) NFE2L2HSD11B1GRIK1GRIK2APP
SCHEMBL8325852 0.78 NFE2L2 (0.45) NFE2L2GRIK1GRIK2TAAR1PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023076218-A1 SPIROTRICYCLE RIPK1 INHIBITORS AND METHODS OF USES THEREOF MERCK SHARP & DOHME LLC (US) 2023-05-04 WO disclosed
US-5543400-A ANTIBIOTICS ROUSSEL UCLAF (FR) 1996-08-06 US disclosed
EP-0606024-B1 Erythromycin derivatives, their process of preparation and their application as medicaments ROUSSEL UCLAF (FR) 1996-03-20 EP disclosed
EP-0606024-A1 Erythromycin derivatives, their process of preparation and their application as medicaments ROUSSEL UCLAF (FR) 1994-07-13 EP disclosed