SCHEMBL8975598

SCHEMBL8975598

C#COc1ccccc1C(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 4/20 0.42
ATM Q13315 1/20 0.42
ALDH1A1 P00352 6/20 0.41
TSHR P16473 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
HSD17B10 Q99714 1/20 0.41
KDM4E B2RXH2 3/20 0.39
GAA P10253 2/20 0.39
RXRA P19793 1/20 0.39
RXRB P28702 1/20 0.39
RXRG P48443 1/20 0.39
MAPT P10636 2/20 0.38
NISCH Q9Y2I1 1/20 0.38
CA2 P00918 1/20 0.38
BCHE P06276 1/20 0.37
NPSR1 Q6W5P4 3/20 0.36
HTT P42858 2/20 0.36
NAMPT P43490 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3826953 0.81 TDP1 (0.41) TDP1ATMALDH1A1TSHRCYP1A2
SCHEMBL3636639 0.81 TDP1 (0.45) TDP1ATMALDH1A1TSHRCYP1A2
SCHEMBL30003749 0.81 TDP1 (0.41) TDP1ATMALDH1A1TSHRCYP1A2
SCHEMBL6874916 0.81 TDP1 (0.41) TDP1ATMALDH1A1TSHRCYP1A2
SCHEMBL20718950 0.78 RXRA (0.39) TDP1ALDH1A1RXRARXRBRXRG
SCHEMBL127278 0.77 ALDH1A1 (0.48) TDP1ATMALDH1A1TSHRCYP1A2
SCHEMBL30500977 0.77 ALDH1A1 (0.48) TDP1ATMALDH1A1TSHRCYP1A2
SCHEMBL6933536 0.75 ALDH1A1 (0.46) TDP1ATMALDH1A1TSHRCYP1A2
SCHEMBL29771456 0.75 CA2 (0.57) TDP1ATMALDH1A1TSHRCYP1A2
SCHEMBL142899 0.75 CA2 (0.57) TDP1ATMALDH1A1TSHRCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0543919-B1 USE OF HETEROCYCLIC AMINO-ALCOHOL COMPOUNDS IN THE MANUFACTURE OF A MEDICAMENT FOR TREATMENT OF CNS DISEASES SEARLE & CO (US) 1996-04-10 EP claimed