SCHEMBL8976235

SCHEMBL8976235

Cn1c2ccc(Br)cc2c2cccnc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FEN1 P39748 1/20 0.42
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
ALOX15 P16050 1/20 0.41
TSHR P16473 1/20 0.41
HSD17B10 Q99714 1/20 0.41
EGFR P00533 3/20 0.40
DDB1 Q16531 1/20 0.40
CRBN Q96SW2 1/20 0.40
PDE4A P27815 3/20 0.40
SRC P12931 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C19 P33261 1/20 0.39
HTT P42858 1/20 0.39
KCNH2 Q12809 2/20 0.38
ACHE P22303 1/20 0.37
TNKS O95271 1/20 0.36
HRH1 P35367 1/20 0.36
HTR6 P50406 1/20 0.36
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16625723 0.82 MEN1 (0.53) FEN1ALDH1A1HPGDTSHRHSD17B10
SCHEMBL12395945 0.79 FEN1 (0.41) FEN1EGFRDDB1CRBNPDE4A
SCHEMBL280139 0.79 GPR3 (0.58) FEN1ALDH1A1HPGDEGFRSRC
SCHEMBL8975764 0.78 FEN1 (0.40) FEN1ALDH1A1HPGDHSD17B10EGFR
SCHEMBL16625727 0.78 CCNB2 (0.42) FEN1HPGDHSD17B10EGFRSRC
SCHEMBL8976112 0.78 BAZ2B (0.44) ALDH1A1HPGDHSD17B10DDB1CRBN
SCHEMBL18381782 0.78 GPR3 (0.56) FEN1ALDH1A1HPGDEGFRSRC
SCHEMBL17339010 0.77 FEN1 (0.46) FEN1ALDH1A1TSHRDDB1CRBN
SCHEMBL17034477 0.77 DDB1 (0.51) FEN1EGFRDDB1CRBNSRC
SCHEMBL1609990 0.76 FEN1 (0.56) FEN1ALDH1A1HPGDEGFRSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008016184-A1 ALPHA-CARBOLINE DERIVATIVES AND METHODS FOR PREPARATION THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-02-07 WO disclosed
US-5532261-A TREATING STAPHYLOCOCCUS INFECTIONS MERCK & CO., INC. (US) 1996-07-02 US disclosed