SCHEMBL8978388

SCHEMBL8978388

CCNc1nc(C)n(C2CCCCC2)c2ncnc1-2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.37
CYP1A2 P05177 3/20 0.37
CYP2C9 P11712 2/20 0.37
MEN1 O00255 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37
STAT3 P40763 1/20 0.37
KMT2A Q03164 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
AURKA O14965 1/20 0.37
JAK2 O60674 1/20 0.37
PRKCA P17252 1/20 0.37
JAK1 P23458 1/20 0.37
KDR P35968 1/20 0.37
GAA P10253 1/20 0.36
ALOX15 P16050 1/20 0.36
CDK9 P50750 2/20 0.35
CCNT1 O60563 1/20 0.35
HCAR1 Q9BXC0 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL27338760 0.99 ALDH1A1 (0.37) ALDH1A1CYP1A2CYP2C9MEN1CYP3A4
SCHEMBL6156828 0.79 PDE10A (0.45) ALDH1A1CYP1A2CYP2C9MEN1CYP3A4
Hydrochloric Acid SCHEMBL27332647 0.78 PDE10A (0.44) ALDH1A1CYP1A2CYP2C9MEN1CYP3A4
SCHEMBL7749667 0.71 PDE10A (0.48) ALDH1A1CYP1A2CYP2C9CYP2D6CASP1
Hydrochloric Acid SCHEMBL27337722 0.70 PDE10A (0.47) ALDH1A1CYP1A2CYP2C9CYP2D6CASP1
SCHEMBL1388102 0.70 YTHDC1 (0.41) JAK2JAK1MAPK14
SCHEMBL8978330 0.70 YTHDC1 (0.41) ALDH1A1CYP1A2CYP2C9CYP3A4CYP2D6
SCHEMBL7415941 0.69 PDE10A (0.34) ALDH1A1CYP1A2CYP2C9CASP1CASP7
Hydrochloric Acid SCHEMBL7742137 0.69 YTHDC1 (0.40) JAK2JAK1MAPK14
SCHEMBL7739861 0.69 KDM4E (0.35) KDM4EADORA3PDE10AADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1045778-C Novel chemical compounds having PDE-IV inhibition activity EURO CELTIQUE SA (LU) 1999-10-20 CN claimed
CN-1125445-A Novel compounds having P.DE-IV inhibitory activity EURO CELTIQUE SA (LU) 1996-06-26 CN claimed
EP-0705265-A1 NOVEL CHEMICAL COMPOUNDS HAVING PDE-IV INHIBITION ACTIVITY Euroceltique S.A. (LU) 1996-04-10 EP claimed
CN-1377353-A Purine derivatives having phosphodiesterase IN inhibition activity EURO CELTIQUE SA (LU) 2002-10-30 CN disclosed