SCHEMBL8979678

SCHEMBL8979678

CNC(=O)CCc1ccc(F)cc1F

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MPO P05164 1/20 0.53
MAOB P27338 1/20 0.46
POLB P06746 1/20 0.46
RAB9A P51151 1/20 0.46
MTNR1A P48039 1/20 0.45
GSK3B P49841 1/20 0.42
BACE1 P56817 1/20 0.42
HDAC1 Q13547 2/20 0.41
HDAC7 Q8WUI4 1/20 0.41
RIPK1 Q13546 2/20 0.41
P2RX7 Q99572 2/20 0.41
DAO P14920 1/20 0.41
CHRNA7 P36544 1/20 0.41
MAPK8 P45983 1/20 0.41
FFAR1 O14842 3/20 0.40
FFAR4 Q5NUL3 2/20 0.40
TP53 P04637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8027585 0.87 MPO (0.50) MPOPOLBRAB9AMTNR1ARIPK1
SCHEMBL13329783 0.83 MAPK8 (0.52) MPOMAOBRIPK1P2RX7MAPK8
SCHEMBL3316261 0.83 MTNR1A (0.61) POLBMTNR1ACHRNA7FFAR1
SCHEMBL30488619 0.81 MAOB (0.53) MAOBGSK3BBACE1RIPK1DAO
SCHEMBL21222818 0.81 MAOB (0.53) MAOBGSK3BBACE1RIPK1DAO
SCHEMBL3576683 0.80 MAOB (0.47) MPOMAOBGSK3BBACE1RIPK1
SCHEMBL20609634 0.80 MAOB (0.49) MAOBPOLBRAB9AGSK3BBACE1
SCHEMBL12851277 0.79 TAAR1 (0.55) MAOBRAB9AMTNR1ARIPK1
SCHEMBL30637597 0.79 FFAR1 (0.59) MAOBPOLBFFAR1FFAR4
SCHEMBL2397247 0.79 FFAR1 (0.59) MAOBPOLBFFAR1FFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5512594-A ADMINISTERING TO TREAT A MEDICAL CONDITION MEDIATED BY ONE OR MORE LEUKOTRIENES ZENECA LIMITED (GB) 1996-04-30 US disclosed
WO-1994025453-A1 4-ARYL-4-HYDROXY-TETRAHYDROPYRANS AND 3-ARYL-3-HYDROXY-TETRAHYDROFURANS AS 5-LIPOXYGENASE INHIBITORS ZENECA LIMITED (GB) 1994-11-10 WO disclosed