SCHEMBL8980367

SCHEMBL8980367

CC(=O)c1cc(NC(=O)c2ccccc2)ccc1N

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.60
POLB P06746 2/20 0.60
HDAC2 Q92769 3/20 0.59
HDAC3 O15379 1/20 0.59
BRAF P15056 1/20 0.59
HDAC4 P56524 1/20 0.59
HDAC1 Q13547 1/20 0.59
HDAC7 Q8WUI4 1/20 0.59
HDAC10 Q969S8 1/20 0.59
HDAC11 Q96DB2 1/20 0.59
HDAC8 Q9BY41 1/20 0.59
HDAC6 Q9UBN7 1/20 0.59
HDAC9 Q9UKV0 1/20 0.59
HDAC5 Q9UQL6 1/20 0.59
KCNK3 O14649 2/20 0.57
KCNK9 Q9NPC2 2/20 0.57
CACNA1B Q00975 1/20 0.57
APBA1 Q02410 1/20 0.57
NPC1 O15118 5/20 0.55
RAB9A P51151 5/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10346126 0.89 KMT2A (0.65) KMT2APOLBHDAC2HDAC3BRAF
SCHEMBL11574206 0.87 HDAC2 (0.53) KMT2APOLBHDAC2HDAC3BRAF
SCHEMBL4409156 0.83 KCNK3 (0.65) KMT2APOLBHDAC2HDAC3HDAC1
SCHEMBL6346820 0.83 KMT2A (0.65) KMT2APOLBKCNK3KCNK9CACNA1B
SCHEMBL3530325 0.83 KMT2A (0.69) KMT2APOLBKCNK3KCNK9CACNA1B
SCHEMBL8980390 0.82 ALDH1A1 (0.53) KMT2APOLBHDAC1NPC1RAB9A
SCHEMBL8278418 0.81 NPC1 (0.71) KMT2APOLBKCNK3KCNK9CACNA1B
SCHEMBL11322912 0.79 RAB9A (0.73) KMT2APOLBKCNK3KCNK9NPC1
SCHEMBL30017323 0.79 NPC1 (0.73) KMT2APOLBHDAC2HDAC3HDAC1
SCHEMBL21473657 0.79 NPC1 (0.73) KMT2APOLBHDAC2HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5571822-A AMINO-2-PHENYL-4-QUINOLONE DERIVATIVES THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1996-11-05 US disclosed
WO-1996010563-A1 2-ARYL-4-QUINOLONES AS ANTITUMOR COMPOUNDS THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1996-04-11 WO disclosed