SCHEMBL8980476

SCHEMBL8980476

COc1ccc(CC(=O)[S])cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.63
SMN1; SMN2 Q16637 3/20 0.58
CTBP2 P56545 1/20 0.56
TDP1 Q9NUW8 2/20 0.54
LDHA P00338 1/20 0.53
KDM4E B2RXH2 2/20 0.53
ALDH1A1 P00352 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2C19 P33261 1/20 0.53
USP2 O75604 1/20 0.53
TP53 P04637 1/20 0.53
POLB P06746 1/20 0.53
F2RL1 P55085 1/20 0.52
MAPT P10636 1/20 0.51
NPC1 O15118 1/20 0.51
PKM P14618 1/20 0.51
LMNA P02545 1/20 0.51
KMT2A Q03164 1/20 0.50
ATM Q13315 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3628705 0.83 HTT (0.68) HTTSMN1; SMN2CTBP2TDP1LDHA
SCHEMBL240822 0.81 KDM4E (0.74) HTTSMN1; SMN2CTBP2TDP1LDHA
SCHEMBL1525068 0.81 HTT (0.66) HTTSMN1; SMN2CTBP2TDP1LDHA
SCHEMBL48525 0.81 HTT (0.66) HTTSMN1; SMN2CTBP2LDHAKDM4E
SCHEMBL28709451 0.81 HTT (0.66) HTTSMN1; SMN2CTBP2LDHAKDM4E
SCHEMBL5257976 0.79 HTT (0.63) HTTSMN1; SMN2CTBP2TDP1LDHA
SCHEMBL3231393 0.79 HTT (0.63) HTTSMN1; SMN2CTBP2TDP1LDHA
SCHEMBL3649876 0.79 HTT (0.63) HTTSMN1; SMN2CTBP2TDP1LDHA
SCHEMBL226124 0.79 HTT (0.63) HTTSMN1; SMN2CTBP2TDP1LDHA
SCHEMBL1067193 0.79 HTT (0.63) HTTSMN1; SMN2CTBP2ALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5519051-A AROMATASE INHIBITORS USEFUL FOR TREATMENT OF DISEASES CAUSED BY EXCESS OF ESTROGEN, FOR EXAMPLE, BREAST CANCER, UTERINE CANCER TEIKOKU HORMONE MFG. CO., LTD. (JP) 1996-05-21 US disclosed
EP-0582713-A1 NOVEL OXA- OR AZASTEROID DERIVATIVE TEIKOKU HORMONE MFG. CO., LTD. (JP) 1994-02-16 EP disclosed