SCHEMBL8980945

SCHEMBL8980945

c1ccn(-c2ccc(Cc3c[nH]nn3)cc2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VHL P40337 1/20 0.44
ELOC Q15369 1/20 0.44
ELOB Q15370 1/20 0.44
POLB P06746 3/20 0.40
NSD2 O96028 1/20 0.40
GRK2 P25098 1/20 0.40
CASP6 P55212 1/20 0.40
CTDSP1 Q9GZU7 1/20 0.40
SMN1; SMN2 Q16637 5/20 0.38
HSD17B10 Q99714 3/20 0.38
LMNA P02545 3/20 0.38
TSHR P16473 2/20 0.38
THRB P10828 1/20 0.38
AOC2 O75106 3/20 0.36
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
MAPK1 P28482 1/20 0.35
MEN1 O00255 5/20 0.34
KMT2A Q03164 5/20 0.34
ALDH1A1 P00352 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29272 0.77 ALDH1A1 (0.46) POLBSMN1; SMN2LMNATSHRRAB9A
Benzene SCHEMBL27499662 0.77 ALDH1A1 (0.46) POLBSMN1; SMN2LMNATSHRRAB9A
SCHEMBL9508013 0.75 ALDH1A1 (0.44) POLBSMN1; SMN2LMNATSHRRAB9A
SCHEMBL20319186 0.74 VHL (0.67) VHLELOCELOBPOLBNSD2
SCHEMBL6944017 0.74 CYP3A4 (0.48) POLBSMN1; SMN2LMNATSHRNPC1
SCHEMBL28117639 0.74 ESR1 (0.48)
SCHEMBL27034778 0.71 ALDH1A1 (0.37) SMN1; SMN2HSD17B10LMNARAB9AKMT2A
SCHEMBL28326701 0.71 HTR1D (0.45) SMN1; SMN2NPC1RAB9AKDM4EHPGD
SCHEMBL3918469 0.71 LTA4H (0.48) POLBSMN1; SMN2LMNARAB9AMEN1
SCHEMBL1818072 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5484937-A ANGIOTENSIN ANTAGONISTS G.D. SEARLE & CO. (US) 1996-01-16 US disclosed
US-5484937-A ANGIOTENSIN ANTAGONISTS G.D. SEARLE & CO. (US) 1996-01-16 US disclosed
US-5484937-A ANGIOTENSIN ANTAGONISTS G.D. SEARLE & CO. (US) 1996-01-16 US disclosed
US-5175180-A Antagonist, antagonism G. D. SEARLE & CO. (US) 1992-12-29 US disclosed
US-5175180-A Antagonist, antagonism G. D. SEARLE & CO. (US) 1992-12-29 US disclosed
WO-1992011255-A1 N-SUBSTITUTED N-(α-TRIAZOLYL-TOLUYL)PYRROLE COMPOUNDS FOR TREATMENT OF CIRCULATORY DISORDERS G.D. SEARLE & CO. (US) 1992-07-09 WO disclosed
WO-1992011255-A1 N-SUBSTITUTED N-(α-TRIAZOLYL-TOLUYL)PYRROLE COMPOUNDS FOR TREATMENT OF CIRCULATORY DISORDERS G.D. SEARLE & CO. (US) 1992-07-09 WO disclosed