Bromide

Bromide

SCHEMBL8987442

Br.NC(=O)c1ccccc1C(=O)NCCCBr.c1ccc(P(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.47

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.47
TSHR P16473 2/20 0.47
NLRP3 Q96P20 1/20 0.42
HPGD P15428 4/20 0.41
NPC1 O15118 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
HSD17B10 Q99714 1/20 0.41
NLRP1 Q9C000 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
POLB P06746 1/20 0.39
ALOX5 P09917 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL308733 0.89 HTT (0.57) HTTTSHRNLRP3HPGDNPC1
SCHEMBL30415135 0.89 HTT (0.57) HTTTSHRNLRP3HPGDNPC1
SCHEMBL2778140 0.84 HTT (0.56) HTTTSHRNLRP3HPGDNPC1
SCHEMBL16487383 0.83 TSHR (0.54) HTTTSHRNLRP3HPGDALOX5
SCHEMBL16486722 0.83 TSHR (0.54) HTTTSHRNLRP3HPGDALOX5
SCHEMBL2080518 0.80 TSHR (0.51) HTTTSHRNLRP3HPGDALDH1A1
SCHEMBL21434178 0.77 LMNA (0.48) TSHRNPC1ALDH1A1MAPTSMN1; SMN2
SCHEMBL6903284 0.76 TSHR (0.58) HTTTSHRHPGDNPC1ALDH1A1
SCHEMBL7255678 0.75 HTT (0.62) HTTTSHRHPGDNPC1ALDH1A1
SCHEMBL9518458 0.74 HTT (0.57) HTTTSHRHPGDNPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5543400-A ANTIBIOTICS ROUSSEL UCLAF (FR) 1996-08-06 US disclosed