SCHEMBL8988263

SCHEMBL8988263

COC(=S)CC(=O)C(F)(F)F

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FAAH O00519 8/20 0.37
CES1 P23141 6/20 0.35
CES2 O00748 5/20 0.35
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35
KMT2A Q03164 1/20 0.35
HSD17B10 Q99714 1/20 0.35
PLOD2 O00469 2/20 0.35
PLOD3 O60568 1/20 0.34
PLOD1 Q02809 1/20 0.34
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL197340 0.75 MGAM (0.48) FAAHCES1CES2MEN1CYP1A2
SCHEMBL17090712 0.75 FAAH (0.39) FAAHCES1CES2MEN1CYP1A2
SCHEMBL183178 0.73 PLOD2 (0.46) FAAHCES1CES2MEN1CYP1A2
SCHEMBL6559914 0.72 PLOD2 (0.39) FAAHCES1CES2MEN1CYP1A2
SCHEMBL6874096 0.72 FAAH (0.41) FAAHCES1CES2MEN1CYP1A2
SCHEMBL28639648 0.72 FAAH (0.41) FAAHCES1CES2MEN1CYP1A2
SCHEMBL17090713 0.71 FAAH (0.37) FAAHCES1CES2MEN1CYP1A2
SCHEMBL9286605 0.71 MAPT (0.36) MEN1KMT2AHSD17B10PLOD2ALDH1A1
Water SCHEMBL7191917 0.70 PLOD2 (0.44) FAAHCES1CES2MEN1CYP1A2
SCHEMBL9283764 0.70 PLOD2 (0.44) FAAHCES1CES2MEN1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0448544-B1 Process for preparation of fluoromethyl-substituted piperidine carbodithioates ROHM & HAAS (US) 1996-07-03 EP claimed
EP-0448544-A2 Process for preparation of fluoromethyl-substituted piperidine carbodithioates ROHM AND HAAS COMPANY (US) 1991-09-25 EP claimed
US-4785129-A Methyl 4,4,4-trifluoro-3-oxo-butanethioate MONSANTO COMPANY (US) 1988-11-15 US claimed
EP-3684352-A1 VANADYL AND VANADATE FOR USE IN REDUCING STRESS -INDUCED METABOLIC DERANGEMENT CFM Pharma Holding BV (NL) 2020-07-29 EP disclosed
WO-2019059770-A1 VANADYL AND VANADATE FOR USE IN REDUCING STRESS -INDUCED METABOLIC DERANGEMENT CFM PHARMA HOLDING B.V. (NL) 2019-03-28 WO disclosed
EP-3412654-A1 PROCESSES FOR THE MANUFACTURE OF HALOALKYL PYRIMIDYL COMPOUNDS, AND COMPOUNDS USEFUL IN THEIR MANUFACTURE SOLVAY SA (BE) 2018-12-12 EP disclosed
EP-3412655-A1 PROCESSES FOR THE MANUFACTURE OF HALOALKYL PYRIMIDYL COMPOUNDS, AND COMPOUNDS USEFUL IN THEIR MANUFACTURE SOLVAY SA (BE) 2018-12-12 EP disclosed
EP-0448544-B1 Process for preparation of fluoromethyl-substituted piperidine carbodithioates ROHM & HAAS (US) 1996-07-03 EP disclosed
EP-0448543-B1 Process for preparation of fluoromethyl-substituted pyridine carbodithioates ROHM & HAAS (US) 1995-12-06 EP disclosed
EP-0448541-B1 Process for preparation of fluoromethyl-substituted pyridine carbodithioates ROHM & HAAS (US) 1995-11-22 EP disclosed
EP-0448542-B1 Process for preparation of fluoromethyl-substituted dihydropyridine carbodithioates ROHM & HAAS (US) 1995-11-22 EP disclosed
US-5099023-A Dehydrofluorination MONSANTO COMPANY (US) 1992-03-24 US disclosed
US-5055583-A Reactive contact with catalytic 1,2-diazabicyclo(2.2.2)octane, salt formation; dehydrohalogenation MONSANTO COMPANY (US) 1991-10-08 US disclosed
EP-0448541-A2 Process for preparation of fluoromethyl-substituted pyridine carbodithioates ROHM AND HAAS COMPANY (US) 1991-09-25 EP disclosed
EP-0448543-A2 Process for preparation of fluoromethyl-substituted pyridine carbodithioates ROHM AND HAAS COMPANY (US) 1991-09-25 EP disclosed
EP-0448544-A2 Process for preparation of fluoromethyl-substituted piperidine carbodithioates ROHM AND HAAS COMPANY (US) 1991-09-25 EP disclosed
EP-0448542-A2 Process for preparation of fluoromethyl-substituted dihydropyridine carbodithioates ROHM AND HAAS COMPANY (US) 1991-09-25 EP disclosed
US-5051512-A Reaction of trifluoroacetic acid thiomethyl ester and ammonia, reaction with an alkyl aldehyde and heating MONSANTO COMPANY (US) 1991-09-24 US disclosed
US-4785129-A Methyl 4,4,4-trifluoro-3-oxo-butanethioate MONSANTO COMPANY (US) 1988-11-15 US disclosed
US-4785129-A Methyl 4,4,4-trifluoro-3-oxo-butanethioate MONSANTO COMPANY (US) 1988-11-15 US disclosed