SCHEMBL8990620

SCHEMBL8990620

CNC(=O)Cc1ccc(N)c(I)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PCNA P12004 2/20 0.48
GAA P10253 4/20 0.41
ALDH1A1 P00352 3/20 0.41
KDM4E B2RXH2 2/20 0.41
MAPT P10636 2/20 0.41
HPGD P15428 1/20 0.41
ALOX15 P16050 1/20 0.41
TSHR P16473 1/20 0.41
HSD17B10 Q99714 1/20 0.41
GFER P55789 1/20 0.41
CDC25B P30305 1/20 0.39
CASP6 P55212 1/20 0.39
RCE1 Q9Y256 1/20 0.39
KLKB1 P03952 1/20 0.38
KMT2A Q03164 2/20 0.38
LMNA P02545 1/20 0.37
ADORA3 P0DMS8 2/20 0.36
HDAC4 P56524 1/20 0.36
CA1 P00915 2/20 0.36
CA2 P00918 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29902856 0.84 GAA (0.47) PCNAGAAALDH1A1KDM4EMAPT
SCHEMBL10663556 0.84 GAA (0.47) PCNAGAAALDH1A1KDM4EMAPT
SCHEMBL5089874 0.81 GAA (0.58) PCNAGAAALDH1A1KDM4EMAPT
SCHEMBL16042637 0.80 ALDH1A1 (0.41) GAAALDH1A1KDM4EMAPTHPGD
SCHEMBL7974514 0.80 ALDH1A1 (0.64) GAAALDH1A1KDM4EMAPTHPGD
SCHEMBL29809190 0.80 ALDH1A1 (0.41) GAAALDH1A1KDM4EMAPTHPGD
SCHEMBL2729682 0.79 HPGD (0.50) PCNAGAAALDH1A1KDM4EMAPT
SCHEMBL10665226 0.75 LMNA (0.49) ALDH1A1MAPTALOX15TSHRKMT2A
SCHEMBL1632446 0.74 LMNA (0.51) ALDH1A1HPGDTSHRGFERKMT2A
SCHEMBL18307178 0.74 LMNA (0.47) PCNAGAAALDH1A1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5583149-A TREATING VASCULAR HEADACHES BRISTOL-MYERS SQUIBB COMPANY (US) 1996-12-10 US disclosed
US-5468768-A FOR TREATING VASCULAR HEADACHES BRISTOL-MYERS SQUIBB COMPANY (US) 1995-11-21 US disclosed
EP-0666258-A1 Indolylcycloaklanylamin- und Indolylcycloalkenylamine derivatives, their preparation and their use as anti-migraine agents Bristol-Myers Squibb Company (US) 1995-08-09 EP disclosed