SCHEMBL8990844

SCHEMBL8990844

Cc1nc(N)c2nc(-c3ccco3)oc2n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 8/20 0.43
KDM4E B2RXH2 7/20 0.43
ALDH1A1 P00352 7/20 0.43
HPGD P15428 6/20 0.43
HSD17B10 Q99714 6/20 0.43
NPC1 O15118 1/20 0.43
CASP3 P42574 1/20 0.43
RAB9A P51151 1/20 0.43
SENP7 Q9BQF6 1/20 0.43
SENP6 Q9GZR1 1/20 0.43
ALOX5 P09917 1/20 0.42
ADORA1 P30542 6/20 0.42
GAA P10253 2/20 0.42
DHFR P00374 1/20 0.41
ADORA3 P0DMS8 4/20 0.41
ADORA2B P29275 3/20 0.40
KMT2A Q03164 1/20 0.39
ELANE P08246 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8990609 0.82 KDM4E (0.45) ADORA2AKDM4EALDH1A1HPGDHSD17B10
SCHEMBL8990648 0.78 KDM4E (0.52) ADORA2AKDM4EALDH1A1HPGDHSD17B10
SCHEMBL8990569 0.77 RAB9A (0.48) KDM4EALDH1A1HPGDHSD17B10NPC1
SCHEMBL1829261 0.76 KDM4E (0.48) KDM4EALDH1A1HPGDHSD17B10NPC1
SCHEMBL8990861 0.75 KDM4E (0.43) ADORA2AKDM4EALDH1A1HPGDHSD17B10
SCHEMBL660601 0.74 KDM4E (0.53) ADORA2AKDM4EALDH1A1HPGDHSD17B10
SCHEMBL660603 0.73 ADORA2A (0.43) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL8990571 0.73 ADK (0.44) ADORA2AKDM4EALDH1A1HPGDHSD17B10
SCHEMBL11838487 0.68 ALDH1A1 (0.57) ADORA2AKDM4EALDH1A1HPGDHSD17B10
SCHEMBL27307267 0.68 ADORA2A (0.48) ADORA2AKDM4EALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5500428-A Furyl-substituted purines and adenosine antagonists IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1996-03-19 US disclosed
US-5300509-A Adenosine antagonists for treating cardiovascular disorders, vasodilation IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1994-04-05 US disclosed
EP-0544445-A2 Furyl-substituted purines, oxazolopyrimidines and pteridines as adenosine antagonists ZENECA LIMITED (GB) 1993-06-02 EP disclosed