SCHEMBL899088

SCHEMBL899088

Fc1cc(Br)ccc1-c1nc2ccc(C(F)(F)F)cc2[nH]1

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NPBWR1 P48145 10/20 0.56
DGAT1 O75907 5/20 0.53
KCNH2 Q12809 5/20 0.53
CBFB Q13951 1/20 0.51
AMY1A P0DUB6 3/20 0.50
SOAT1 P35610 2/20 0.49
FGFR1 P11362 1/20 0.46
FLT3 P36888 1/20 0.46
CLK4 Q9HAZ1 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15231839 0.90 NPBWR1 (0.43) NPBWR1DGAT1KCNH2CBFBAMY1A
SCHEMBL900794 0.81 NPBWR1 (0.74) NPBWR1DGAT1KCNH2CBFBSOAT1
SCHEMBL2898110 0.79 NPC1 (0.67) AMY1AFGFR1
SCHEMBL18229694 0.77 HDAC6 (0.66)
SCHEMBL27040014 0.77 NPBWR1 (0.72) NPBWR1DGAT1KCNH2CBFBSOAT1
SCHEMBL31593060 0.77 NPBWR1 (0.72) NPBWR1DGAT1KCNH2CBFBSOAT1
SCHEMBL4176876 0.77 CBFB (0.71) NPBWR1DGAT1KCNH2CBFBSOAT1
SCHEMBL10325798 0.76 NPBWR1 (0.64) NPBWR1DGAT1KCNH2CBFBSOAT1
SCHEMBL26597176 0.76 ALDH1A1 (0.67) AMY1A
SCHEMBL14074150 0.76 DYRK1A (0.57) NPBWR1DGAT1KCNH2CBFBSOAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013130370-A2 COMPOUNDS AS DGAT-1 INHIBITORS MERCK SHARP & DOHME CORP. (US) 2013-09-06 WO disclosed
WO-2013130370-A2 COMPOUNDS AS DGAT-1 INHIBITORS MERCK SHARP & DOHME CORP. (US) 2013-09-06 WO disclosed
WO-2012096813-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-07-19 WO disclosed
WO-2012044567-A2 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed