SCHEMBL8991819

SCHEMBL8991819

S=C1[N]c2ccccc2N1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MAPT P10636 8/20 0.35
MEN1 O00255 6/20 0.35
KMT2A Q03164 6/20 0.35
KDM4E B2RXH2 3/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
HSP90AA1 P07900 1/20 0.35
THRB P10828 1/20 0.35
HK1 P19367 1/20 0.35
MAPK1 P28482 1/20 0.35
RECQL P46063 1/20 0.35
GALK1 P51570 1/20 0.35
BLM P54132 1/20 0.35
HKDC1 Q2TB90 1/20 0.35
ALDH1A1 P00352 4/20 0.34
GAA P10253 5/20 0.33
NOX1 Q9Y5S8 2/20 0.33
USP2 O75604 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1236095 1.00 LMNA (0.36) LMNASMN1; SMN2MAPTMEN1KMT2A
SCHEMBL240371 0.79 MAPT (0.43) LMNASMN1; SMN2MAPTMEN1KMT2A
SCHEMBL9203699 0.77 ALDH1A1 (0.37) LMNASMN1; SMN2MAPTMEN1KMT2A
SCHEMBL9204546 0.73 ALDH1A1 (0.37) LMNASMN1; SMN2KDM4EALDH1A1PPARG
SCHEMBL2475507 0.71 LMNA (0.36) LMNASMN1; SMN2MAPTMEN1KMT2A
SCHEMBL20723 0.71 MAPT (0.44) LMNASMN1; SMN2MAPTMEN1KMT2A
SCHEMBL20505096 0.71 MAPT (0.44) LMNASMN1; SMN2MAPTMEN1KMT2A
SCHEMBL3541281 0.70 GSK3B (0.48) LMNASMN1; SMN2MAPTMEN1KMT2A
SCHEMBL13819803 0.69 MAPT (0.43) LMNASMN1; SMN2MAPTMEN1KMT2A
SCHEMBL554552 0.68 MAPT (0.46) LMNASMN1; SMN2MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0465254-B1 Fused thiophene compounds and uses thereof YOSHITOMI PHARMACEUTICAL (JP) 1996-11-13 EP claimed
US-5141930-A Antianxietic drug, antipsychotics and cardiotonic agents YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1992-08-25 US claimed
EP-0465254-B1 Fused thiophene compounds and uses thereof YOSHITOMI PHARMACEUTICAL (JP) 1996-11-13 EP disclosed
US-5532240-A ANTIPSYCHOTIC AGENTS AND ANTISEROTONIN AGENTS YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1996-07-02 US disclosed
US-5466691-A Antipsychotic and anxiolytic agents YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1995-11-14 US disclosed
EP-0596120-A1 THIOPHENE COMPOUND YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1994-05-11 EP disclosed
EP-0596125-A1 CONDENSED THIOPHENE COMPOUND AND PHARMACEUTICAL USE THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1994-05-11 EP disclosed
US-5141930-A Antianxietic drug, antipsychotics and cardiotonic agents YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1992-08-25 US disclosed
EP-0465254-A1 Fused thiophene compounds and uses thereof YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1992-01-08 EP disclosed