SCHEMBL8992523

SCHEMBL8992523

CCCc1nc(CC#N)c[nH]1

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.32
MAPT P10636 1/20 0.32
KMT2A Q03164 1/20 0.32
CTSK P43235 8/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPK1 P28482 1/20 0.31
CTSS P25774 6/20 0.31
KDM5A P29375 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1985579 0.84 CTSK (0.31) KMT2ACTSKALDH1A1MAPK1CTSS
SCHEMBL28336002 0.83 MEN1 (0.40) MEN1MAPTKMT2A
SCHEMBL3286058 0.81 BACE1 (0.36) MAPTALDH1A1
SCHEMBL3697323 0.79 GLA (0.33)
SCHEMBL8992520 0.76 ADORA3 (0.33)
SCHEMBL9937448 0.76 SMN1; SMN2 (0.32)
SCHEMBL3841860 0.76 HRH3 (0.41) ALDH1A1MAPK1
SCHEMBL9237749 0.73
SCHEMBL8531352 0.73 HRH3 (0.32) MEN1KMT2A
Hydrochloric Acid SCHEMBL8992515 0.73 HRH4 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0531876-B1 Imidazoindolizine derivatives and process for preparation thereof TANABE SEIYAKU CO (JP) 1996-12-18 EP disclosed
US-5510354-A HYPOTENSIVE AGENTS TANABE SEIYAKU CO., LTD. (JP) 1996-04-23 US disclosed
US-5424316-A Imidazopyridine derivatives for the treatment of hypertension TANABE SEIYAKU CO., LTD. (JP) 1995-06-13 US disclosed
US-5409936-A Useful in prophylaxix; exhibits potent angiotensin ii inhibitory acivities TANABE SEIYAKU CO., LTD. (JP) 1995-04-25 US disclosed
US-5268377-A Imidazoindolizine derivatives process for preparation thereof and use thereof to treat hypertension TANABE SEIYAKU CO., LTD. (JP) 1993-12-07 US disclosed
EP-0531876-A2 Imidazoindolizine derivatives and process for preparation thereof TANABE SEIYAKU CO., LTD. (JP) 1993-03-17 EP disclosed
EP-0531874-A1 Imidazopyridine derivatives and process for preparation thereof TANABE SEIYAKU CO., LTD. (JP) 1993-03-17 EP disclosed