SCHEMBL8992953

SCHEMBL8992953

CCOC(=O)c1ccc(C(O)c2ccc(OC)cc2)c(OC)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B2 P37059 1/20 0.56
SMN1; SMN2 Q16637 2/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
TAS1R3 Q7RTX0 1/20 0.45
TAS1R1 Q7RTX1 1/20 0.45
MAPK1 P28482 2/20 0.44
TSHR P16473 2/20 0.44
HSD17B10 Q99714 1/20 0.44
KMT2A Q03164 3/20 0.44
KDM4E B2RXH2 1/20 0.44
POLB P06746 1/20 0.44
MAPT P10636 4/20 0.44
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
MEN1 O00255 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C19 P33261 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8993178 0.91 HSD17B2 (0.57) HSD17B2SMN1; SMN2NPC1RAB9AMAPK1
SCHEMBL8992796 0.83 HSD17B2 (0.59) HSD17B2SMN1; SMN2NPC1RAB9AMAPK1
SCHEMBL8992942 0.80 HSD17B2 (0.56) HSD17B2SMN1; SMN2NPC1RAB9AMAPK1
SCHEMBL4284989 0.79 CA12 (0.55) HSD17B2SMN1; SMN2NPC1RAB9AHSD17B10
SCHEMBL10686479 0.78 LMNA (0.54) NPC1MAPK1KMT2AMAPTALDH1A1
4-Methoxybenzoic Acid Ethyl Ester SCHEMBL203475 0.76 CA1 (0.66) HSD17B2SMN1; SMN2NPC1RAB9AKMT2A
SCHEMBL6929080 0.75 HSD17B2 (0.59) HSD17B2SMN1; SMN2NPC1RAB9AMAPK1
SCHEMBL21469937 0.75 MAPT (0.51) SMN1; SMN2HSD17B10KMT2AMAPTALDH1A1
SCHEMBL30506315 0.75 HSD17B2 (0.76) HSD17B2SMN1; SMN2NPC1RAB9AMAPK1
SCHEMBL1660365 0.75 HSD17B2 (0.76) HSD17B2SMN1; SMN2NPC1RAB9AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516777-A PROSTATE CANCER THERAPY OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-05-14 US disclosed
US-5409928-A Prostate diseases, alopecia OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-04-25 US disclosed
EP-0594149-A2 Condensed pyrazole derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-04-27 EP disclosed