SCHEMBL8992998

SCHEMBL8992998

COc1cccc(Cc2ccc(C=O)cc2)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.54
RAB9A P51151 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
MTNR1A P48039 1/20 0.53
MTNR1B P49286 1/20 0.53
ALDH1A1 P00352 1/20 0.53
CYP2A6 P11509 1/20 0.53
HDAC3 O15379 1/20 0.51
HDAC1 Q13547 1/20 0.51
HDAC2 Q92769 1/20 0.51
HDAC8 Q9BY41 1/20 0.51
LTA4H P09960 3/20 0.50
CHRM2 P08172 2/20 0.50
CHRM1 P11229 2/20 0.50
CHRM3 P20309 2/20 0.50
LMNA P02545 1/20 0.49
TP53 P04637 1/20 0.49
MAPT P10636 1/20 0.49
CMA1 P23946 1/20 0.49
TAAR1 Q96RJ0 3/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27514736 0.90 NPC1 (0.57) NPC1RAB9ATDP1MTNR1AMTNR1B
SCHEMBL18635836 0.86 HDAC1 (0.68) NPC1RAB9ATDP1ALDH1A1HDAC3
Ethylene SCHEMBL8992917 0.85 MTNR1A (0.46) NPC1RAB9ATDP1MTNR1AMTNR1B
SCHEMBL14191204 0.84 LTA4H (0.70) MTNR1AMTNR1BALDH1A1LTA4HCHRM2
SCHEMBL2099512 0.84 CHRM2 (0.66) LTA4HCHRM2CHRM1CHRM3CMA1
SCHEMBL8024555 0.83 NPC1 (0.66) NPC1RAB9ATDP1MTNR1AMTNR1B
SCHEMBL6687219 0.83 MAOB (0.66) NPC1RAB9ATDP1TP53MEN1
SCHEMBL2092574 0.82 LTA4H (0.67) MTNR1AMTNR1BLTA4HCHRM2CHRM1
SCHEMBL9607336 0.82 ALDH1A1 (0.79) NPC1RAB9ATDP1ALDH1A1CYP2A6
SCHEMBL31739258 0.82 LTA4H (0.67) MTNR1AMTNR1BLTA4HCHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed
US-5516777-A PROSTATE CANCER THERAPY OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-05-14 US disclosed
US-5409928-A Prostate diseases, alopecia OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-04-25 US disclosed
EP-0594149-A2 Condensed pyrazole derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-04-27 EP disclosed