SCHEMBL8993065

SCHEMBL8993065

CCOC(=O)CC(=O)N1CCc2nc(CC)n(Cc3ccc(-c4ccccc4C(=O)O)cc3)c2C1C(=O)OCC

nearest known ligand 0.50

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PPARG P37231 2/20 0.42
AGTR1 P30556 1/20 0.42
AGTR2 P50052 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8992476 0.94 PPARG (0.50) PPARG
SCHEMBL9140447 0.91 PPARG (0.44) PPARGAGTR1AGTR2
SCHEMBL9046073 0.91 ACHE (0.43)
SCHEMBL9043822 0.89 PPARG (0.51) PPARG
SCHEMBL9043551 0.86 ACHE (0.48) AGTR1AGTR2
SCHEMBL9045425 0.86 AGTR1 (0.39) PPARGAGTR1AGTR2
SCHEMBL9582592 0.86 PPARG (0.41) PPARGAGTR1AGTR2
SCHEMBL9045308 0.85 ACHE (0.45) PPARG
SCHEMBL9255274 0.81 ACHE (0.43)
SCHEMBL8992556 0.81 PPARG (0.54) PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0531876-B1 Imidazoindolizine derivatives and process for preparation thereof TANABE SEIYAKU CO (JP) 1996-12-18 EP disclosed
US-5510354-A HYPOTENSIVE AGENTS TANABE SEIYAKU CO., LTD. (JP) 1996-04-23 US disclosed
US-5424316-A Imidazopyridine derivatives for the treatment of hypertension TANABE SEIYAKU CO., LTD. (JP) 1995-06-13 US disclosed
US-5409936-A Useful in prophylaxix; exhibits potent angiotensin ii inhibitory acivities TANABE SEIYAKU CO., LTD. (JP) 1995-04-25 US disclosed
US-5268377-A Imidazoindolizine derivatives process for preparation thereof and use thereof to treat hypertension TANABE SEIYAKU CO., LTD. (JP) 1993-12-07 US disclosed
EP-0531876-A2 Imidazoindolizine derivatives and process for preparation thereof TANABE SEIYAKU CO., LTD. (JP) 1993-03-17 EP disclosed
EP-0531874-A1 Imidazopyridine derivatives and process for preparation thereof TANABE SEIYAKU CO., LTD. (JP) 1993-03-17 EP disclosed