SCHEMBL899315

SCHEMBL899315

COc1ccc(Nc2nccs2)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.64
LMNA P02545 2/20 0.64
TP53 P04637 1/20 0.64
TSHR P16473 1/20 0.64
PKM P14618 3/20 0.63
RAB9A P51151 8/20 0.57
NPC1 O15118 6/20 0.57
PTGS2 P35354 2/20 0.56
MAPT P10636 5/20 0.53
GAA P10253 5/20 0.53
RECQL P46063 3/20 0.53
KDM4E B2RXH2 2/20 0.53
TDP1 Q9NUW8 2/20 0.53
THRB P10828 1/20 0.53
MAPK1 P28482 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
MEN1 O00255 5/20 0.52
KMT2A Q03164 5/20 0.52
ALDH1A1 P00352 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9381614 0.87 RAB9A (0.65) SMN1; SMN2LMNATP53TSHRPKM
Water SCHEMBL9387383 0.86 RAB9A (0.64) SMN1; SMN2LMNATP53TSHRPKM
SCHEMBL5706320 0.81 SYK (0.53) SMN1; SMN2LMNATP53TSHRPKM
SCHEMBL3525964 0.81 PKM (0.50) SMN1; SMN2LMNATP53TSHRPKM
SCHEMBL10045058 0.81 CYP1A2 (0.67) SMN1; SMN2TSHRPKMRAB9ANPC1
SCHEMBL5762561 0.80 PLA2G7 (0.58) SMN1; SMN2LMNATP53TSHRPKM
SCHEMBL27791948 0.79 NPC1 (0.50) SMN1; SMN2LMNATP53TSHRPKM
SCHEMBL27431502 0.79 SMN1; SMN2 (0.71) SMN1; SMN2LMNATP53TSHRPKM
SCHEMBL15508074 0.78 PKM (1.00) SMN1; SMN2LMNATSHRPKMGAA
SCHEMBL28717675 0.78 CYP1A2 (0.77) SMN1; SMN2RAB9ANPC1PTGS2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112390755-B Heteroaryl method for amine 中国科学院理化技术研究所 2024-08-02 CN claimed
EP-3812040-B1 COMPLEXES JOHNSON MATTHEY PLC (GB) 2023-01-11 EP disclosed
EP-3812040-B1 COMPLEXES JOHNSON MATTHEY PLC (GB) 2023-01-11 EP disclosed
CN-110201721-B Complex compounds 庄信万丰股份有限公司 2022-07-22 CN disclosed
EP-3812040-A1 COMPLEXES Johnson Matthey Public Limited Company (GB) 2021-04-28 EP disclosed
EP-3812040-A1 COMPLEXES Johnson Matthey Public Limited Company (GB) 2021-04-28 EP disclosed
EP-3154689-B1 COMPLEXES JOHNSON MATTHEY PLC (GB) 2021-01-27 EP disclosed
CN-106661071-B Complex compounds 庄信万丰股份有限公司 2020-06-09 CN disclosed
US-9777030-B2 Complexes JOHNSON MATTHEY PUBLIC LIMITED COMPANY (GB) 2017-10-03 US disclosed
US-9777030-B2 Complexes JOHNSON MATTHEY PUBLIC LIMITED COMPANY (GB) 2017-10-03 US disclosed
WO-2012040754-A2 NOVEL THIAZOLAMINE DERIVATES AS DIFFERENTIATION ACCELERATORS TECHNISCHE UNIVERSITÄT WIEN (AT) 2012-04-05 WO disclosed
WO-2012040754-A2 NOVEL THIAZOLAMINE DERIVATES AS DIFFERENTIATION ACCELERATORS TECHNISCHE UNIVERSITÄT WIEN (AT) 2012-04-05 WO disclosed
US-7795288-B2 Thiazole and pyrazole derivatives as Flt-3 kinase inhibitors NOVARTIS AG (CH) 2010-09-14 US disclosed
US-7795288-B2 Thiazole and pyrazole derivatives as Flt-3 kinase inhibitors NOVARTIS AG (CH) 2010-09-14 US disclosed
US-7795288-B2 Thiazole and pyrazole derivatives as Flt-3 kinase inhibitors NOVARTIS AG (CH) 2010-09-14 US disclosed
US-20070167449-A1 Thiazole and pyrazole derivatives as flt-3 kinase inhibitors NOVARTIS PHARMA AG (CH) 2007-07-19 US disclosed
US-20070167449-A1 Thiazole and pyrazole derivatives as flt-3 kinase inhibitors NOVARTIS PHARMA AG (CH) 2007-07-19 US disclosed
US-20070167449-A1 Thiazole and pyrazole derivatives as flt-3 kinase inhibitors NOVARTIS PHARMA AG (CH) 2007-07-19 US disclosed
EP-1687285-A1 THIAZOLE AND PYRAZOLE DERIVATIVES AS FLT-3 KINASE INHIBITORS Novartis AG (CH) 2006-08-09 EP disclosed
WO-2005047273-A1 THIAZOLE AND PYRAZOLE DERIVATIVES AS FLT-3 KINASE INHIBITORS NOVARTIS AG (CH) 2005-05-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070167449-A1 Thiazole and pyrazole derivatives as flt-3 kinase inhibitors FLT3, FLT1, FLT4 SMN1; SMN2 4364/4885LMNA 2263/4885TP53 130/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.