SCHEMBL8993292

SCHEMBL8993292

CS(=O)(=O)c1ccccc1C(=CC(O)c1ccc(F)cc1)CO

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 1/20 0.35
HTR2A P28223 2/20 0.35
HTR2C P28335 2/20 0.35
KCNH2 Q12809 2/20 0.35
PTGS2 P35354 3/20 0.35
CYP2D6 P10635 2/20 0.34
NAAA Q02083 1/20 0.34
MDM2 Q00987 1/20 0.33
ACLY P53396 1/20 0.33
KAT6A Q92794 3/20 0.33
LMNA P02545 1/20 0.32
EPHX2 P34913 3/20 0.32
CYP3A4 P08684 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8993288 0.77 EPHX2 (0.48) PTGS2EPHX2
SCHEMBL8388365 0.70 ESR2 (0.44) BCAT2PTGS2LMNA
SCHEMBL7614169 0.68 BCAT2 (0.53) BCAT2LMNA
SCHEMBL8388530 0.64 ESR2 (0.40) BCAT2PTGS2LMNA
SCHEMBL800185 0.63 AOC3 (0.40)
SCHEMBL13651738 0.62 BCAT2 (0.53) BCAT2LMNA
SCHEMBL6904881 0.62 PTGS2 (0.68) PTGS2SLC6A4SLC6A3
SCHEMBL30455726 0.61 BCAT2 (0.51) BCAT2LMNA
SCHEMBL5028957 0.61 BCAT2 (0.51) BCAT2LMNA
SCHEMBL4321077 0.61 BCAT2 (0.59) BCAT2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0724566-A1 1,2-DIARYLCYCLOPENTENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-08-07 EP disclosed
WO-1995011883-A1 1,2-DIARYLCYCLOPENTENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-05-04 WO disclosed