SCHEMBL8994033

SCHEMBL8994033

Cn1c(C(N)I)nc(-c2ccccc2)cc1=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.48
BACE1 P56817 3/20 0.43
ADORA1 P30542 1/20 0.43
TP53 P04637 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
KDM4E B2RXH2 2/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
HPGD P15428 1/20 0.43
RAD51 Q06609 1/20 0.43
GSK3B P49841 6/20 0.42
CGAS Q8N884 1/20 0.40
MEN1 O00255 1/20 0.40
MAPT P10636 1/20 0.40
KMT2A Q03164 1/20 0.40
KDM5B Q9UGL1 1/20 0.40
CDC7 O00311 1/20 0.40
ROCK2 O75116 1/20 0.40
MAP4K4 O95819 1/20 0.40
PIM1 P11309 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4493177 0.76 BACE1 (0.63) ALDH1A1BACE1ADORA1TP53SMN1; SMN2
SCHEMBL8767485 0.74 ALDH1A1 (0.56) ALDH1A1BACE1ADORA1TP53SMN1; SMN2
SCHEMBL11502325 0.71 ADORA1 (0.56) ALDH1A1ADORA1TP53SMN1; SMN2KDM4E
SCHEMBL8994051 0.70 GSK3B (0.56) ALDH1A1BACE1ADORA1TP53SMN1; SMN2
SCHEMBL7385338 0.69 GSK3B (0.59) ALDH1A1GSK3BMEN1KMT2ACDC7
SCHEMBL4508981 0.69 BACE1 (0.67) BACE1KDM4E
SCHEMBL10844457 0.67 KDM4E (0.48) ALDH1A1BACE1ADORA1TP53SMN1; SMN2
SCHEMBL4148126 0.66 BACE1 (0.57) ALDH1A1BACE1ADORA1SMN1; SMN2KDM4E
SCHEMBL11665619 0.66 ALDH1A1 (0.49) ALDH1A1ADORA1TP53SMN1; SMN2KDM4E
SCHEMBL11797265 0.65 ALDH1A1 (1.00) ALDH1A1ADORA1TP53SMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0724573-A1 PYRIMIDINONES AS ANTIARTHRITIC AND ANTI-INFLAMMATORIES PHARMACIA & UPJOHN COMPANY (US) 1996-08-07 EP disclosed
WO-1995011235-A1 PYRIMIDINONES AS ANTIARTHRITIC AND ANTI-INFLAMMATORIES THE UPJOHN COMPANY (US) 1995-04-27 WO disclosed