SCHEMBL8994981

SCHEMBL8994981

COc1cc(OCCCCCOc2ccc(C(=O)N(C(C)C)C(C)C)cc2)ccc1C=NN

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTB4R Q15722 3/20 0.57
LTB4R2 Q9NPC1 1/20 0.55
KDM4E B2RXH2 3/20 0.42
ALDH1A1 P00352 2/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
POLB P06746 1/20 0.42
NPY1R P25929 1/20 0.42
NPY2R P49146 1/20 0.42
RAB9A P51151 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
MAOB P27338 2/20 0.41
MAPT P10636 2/20 0.40
PTPN1 P18031 2/20 0.40
CYP1A1 P04798 1/20 0.39
CYP1B1 Q16678 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
LSS P48449 1/20 0.38
HPGD P15428 1/20 0.38
EGFR P00533 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9701994 0.90 LTB4R (0.47) LTB4RLTB4R2KDM4EALDH1A1MEN1
SCHEMBL9117727 0.82 LTB4R (0.52) LTB4RLTB4R2ALDH1A1PLA2G4B
SCHEMBL7711975 0.82 LTB4R (0.72) LTB4RLTB4R2KDM4EALDH1A1POLB
Hydrochloric Acid SCHEMBL8994941 0.82 LTB4R (0.51) LTB4RLTB4R2ALDH1A1PLA2G4B
Hydrochloric Acid SCHEMBL8994890 0.81 LTB4R (0.71) LTB4RLTB4R2KDM4EALDH1A1POLB
Hydrochloric Acid SCHEMBL8995021 0.81 LTB4R (0.68) LTB4RLTB4R2MAPTPLA2G4B
Hydrochloric Acid SCHEMBL8994966 0.81 LTB4R (0.49) LTB4RLTB4R2ALDH1A1MEN1KMT2A
Hydrochloric Acid SCHEMBL8995013 0.80 LTB4R (0.56) LTB4RLTB4R2KDM4EALDH1A1MAOB
SCHEMBL9702013 0.80 LTB4R (0.68) LTB4RLTB4R2KDM4EALDH1A1MEN1
SCHEMBL8994985 0.80 LTB4R (0.68) LTB4RLTB4R2KDM4EALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5488160-A LEUKOTRIENE B4 RECEPTOR ANTAGONIST AS ANTIINFLAMMATORY AGENTS CIBA-GEIGY CORPORATION (US) 1996-01-30 US disclosed
US-5451700-A Leukotriene inhibitors CIBA-GEIGY CORPORATION (US) 1995-09-19 US disclosed
EP-0518819-B1 Amidino compounds, their manufacture and use as medicament CIBA GEIGY AG (CH) 1995-08-02 EP disclosed