SCHEMBL9701994

SCHEMBL9701994

COc1cc(OCCCCCOc2ccc(C(=O)N(C(C)CI)C(C)CI)cc2)ccc1C=NN

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTB4R Q15722 3/20 0.47
LTB4R2 Q9NPC1 1/20 0.45
MAOB P27338 2/20 0.39
KDM4E B2RXH2 3/20 0.38
ALDH1A1 P00352 2/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
POLB P06746 1/20 0.38
NPY1R P25929 1/20 0.38
NPY2R P49146 1/20 0.38
RAB9A P51151 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MAPT P10636 2/20 0.38
PTPN1 P18031 2/20 0.38
GAA P10253 1/20 0.38
CYP1A1 P04798 1/20 0.37
CYP1B1 Q16678 1/20 0.37
LSS P48449 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
GPR119 Q8TDV5 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8994981 0.90 LTB4R (0.57) LTB4RLTB4R2MAOBKDM4EALDH1A1
SCHEMBL9699613 0.83 LTB4R (0.59) LTB4RLTB4R2MAOBKDM4EALDH1A1
Hydrochloric Acid SCHEMBL9701746 0.83 GAA (0.43) LTB4RLTB4R2MAOBALDH1A1GAA
Hydrochloric Acid SCHEMBL9701722 0.83 LTB4R (0.58) LTB4RLTB4R2MAOBKDM4EALDH1A1
Hydrochloric Acid SCHEMBL9700771 0.82 THRA (0.41) LTB4RLTB4R2MAOBMAPTLSS
Hydrochloric Acid SCHEMBL9700974 0.81 LTB4R (0.46) LTB4RLTB4R2MAPTGAAHDAC8
Hydrochloric Acid SCHEMBL9701752 0.78 LTB4R (0.39) LTB4RLTB4R2ALDH1A1MAPTHDAC8
Hydrochloric Acid SCHEMBL9701749 0.76 THRA (0.39) LTB4RLTB4R2MAOBNPSR1MAPT
SCHEMBL9700776 0.76 LTB4R (0.37) LTB4RLTB4R2GAALSSHDAC8
Hydrochloric Acid SCHEMBL9700781 0.75 LTB4R (0.36) LTB4RLTB4R2MAPTGAAGPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0518819-A2 Amidino compounds, their manufacture and use as medicament CIBA-GEIGY AG (CH) 1992-12-16 EP disclosed