SCHEMBL8995844

SCHEMBL8995844

Nc1nc(O)cc(-c2cccc(Cl)c2)n1

nearest known ligand 0.71

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 2/20 0.52
HRH4 Q9H3N8 1/20 0.51
ADORA2A P29274 6/20 0.49
ADORA1 P30542 6/20 0.49
ADORA2B P29275 2/20 0.49
KDM4E B2RXH2 1/20 0.49
HSP90AA1 P07900 1/20 0.49
HSP90AB1 P08238 1/20 0.49
ATP4A P20648 2/20 0.48
ATP4B P51164 2/20 0.48
DHFR P00374 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4277540 0.83 HSP90AA1 (0.71) MAP4K4HRH4ADORA2AADORA1ADORA2B
SCHEMBL7383081 0.83 ATP4A (0.47) ATP4AATP4B
SCHEMBL18931741 0.81 KDM4E (0.58) HRH4ADORA2AADORA1KDM4EHSP90AA1
SCHEMBL3451102 0.80 ADORA2A (0.73) HRH4ADORA2AADORA1KDM4EHSP90AA1
SCHEMBL5747382 0.80 HSP90AA1 (0.58) MAP4K4HRH4ADORA2AADORA1ADORA2B
SCHEMBL19762220 0.77 MEN1 (0.50) ADORA2AADORA1KDM4E
SCHEMBL2324638 0.73 ADORA2A (0.53) MAP4K4HRH4ADORA2AADORA1ADORA2B
SCHEMBL14413006 0.73 HSP90AA1 (0.67) MAP4K4HRH4ADORA2AADORA1ADORA2B
SCHEMBL15757436 0.73 HRH4 (0.57) MAP4K4HRH4ADORA2AADORA1ADORA2B
SCHEMBL9566496 0.73 RAB9A (0.61) MAP4K4HRH4ADORA2AADORA1ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5554617-A Method for treating cancer with 6-aryl pyrimidine compounds THE UPJOHN COMPANY (US) 1996-09-10 US disclosed
US-5434157-A Active against herpes, hepatitis, papovavirus THE UPJOHN COMPANY (US) 1995-07-18 US disclosed
US-5002951-A 2-amino-5-halo-4-pyrimidinol for bactericides and antiprotozoa agent THE UPJOHN COMPANY (US) 1991-03-26 US disclosed
US-4665077-A IMMUNOREGULATORY AGENTS THE UPJOHN COMPANY (US) 1987-05-12 US disclosed
US-4619933-A 6-aryl pyrimidines for treating aplastic anemia THE UPJOHN COMPANY (US) 1986-10-28 US disclosed
US-4543248-A Method for immunoregulation with 6-aryl pyrimidine compounds THE UPJOHN COMPANY (US) 1985-09-24 US disclosed
US-4507302-A Method for treating arthritis with 6-aryl pyrimidine compounds THE UPJOHN COMPANY (US) 1985-03-26 US disclosed