SCHEMBL8995969

SCHEMBL8995969

Cn1ncnc1C(=O)NC1CC1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.43
SMYD3 Q9H7B4 3/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
KDM4E B2RXH2 1/20 0.42
HTT P42858 1/20 0.42
ALDH1A1 P00352 1/20 0.41
PDE4B Q07343 5/20 0.41
KAT2B Q92831 1/20 0.40
CNR1 P21554 1/20 0.39
PDE4D Q08499 1/20 0.39
LMNA P02545 1/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21490096 0.93 SMYD3 (0.55) SMYD3
SCHEMBL19710530 0.93 SMYD3 (0.55) SMYD3
SCHEMBL8950348 0.80 HTR4 (0.41) SMYD3SMN1; SMN2L3MBTL1KDM4EHTT
SCHEMBL12495652 0.77 BAZ2B (0.42) SMN1; SMN2KDM4EHTTALDH1A1LMNA
SCHEMBL2214845 0.70
SCHEMBL19710187 0.69 SMYD3 (0.50) SMYD3
SCHEMBL21490181 0.69 SMYD3 (0.50) SMYD3
SCHEMBL12851851 0.69 CNR1 (0.42) HPGDSMYD3KDM4EHTTPDE4B
SCHEMBL10364892 0.69 HSD11B1 (0.52) HPGDSMN1; SMN2KDM4EHTTALDH1A1
SCHEMBL12496155 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8188085-B2 Antifungal agents MERCK SHARP & DOHME CORP. (US) 2012-05-29 US disclosed
US-20100113439-A1 Antifungal agents MERCK & CO., INC. (US) 2010-05-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100113439-A1 Antifungal agents GMDS, GBA3, UGGT1 HPGD 413/4885SMYD3 3041/4885SMN1; SMN2 3768/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.