SCHEMBL8997147

SCHEMBL8997147

CC(C)(C)OC(=O)c1ccc(CCCc2c[nH]c3nc(N)nc(N)c23)cc1

nearest known ligand 0.60

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.50
DHFR P00374 4/20 0.43
TYMS P04818 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9085311 0.89 NAMPT (0.53) NAMPTDHFRTYMS
SCHEMBL9044536 0.87 NAMPT (0.51) NAMPTDHFRTYMS
SCHEMBL7836419 0.84 NAMPT (0.56) NAMPTDHFRTYMS
SCHEMBL8997200 0.83 NAMPT (0.42) NAMPTDHFRTYMS
SCHEMBL9431448 0.82 NAMPT (0.53) NAMPTDHFRTYMS
SCHEMBL9439883 0.81 FOLR1 (0.44) NAMPT
SCHEMBL8997197 0.81 DHFR (0.37) NAMPTDHFRTYMS
SCHEMBL7843188 0.80 NAMPT (0.57) NAMPTDHFRTYMS
SCHEMBL8982456 0.80 CYP4A11 (0.48) NAMPTDHFRTYMS
SCHEMBL8982532 0.79 CYP4A11 (0.45) NAMPTDHFRTYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0334636-B1 Pyrrolopyrimidine derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1996-10-23 EP disclosed
US-5539113-A ANTITUMOR AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-07-23 US disclosed
US-5496946-A Production of pyrrolopyrimidines and intermediates therefor TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-03-05 US disclosed
US-5349064-A Production of pyrrolopyrimidines TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-09-20 US disclosed
US-5296600-A Antitumor agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-03-22 US disclosed
US-5106974-A Antitumor and -carcinogenic agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-04-21 US disclosed
US-4997838-A Antitumor agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1991-03-05 US disclosed
EP-0402903-A1 Production of pyrrolopyrimidines and intermediates therefor Takeda Chemical Industries, Ltd. (JP) 1990-12-19 EP disclosed