SCHEMBL8997197

SCHEMBL8997197

CC(C)(C)OC(=O)c1ccc(CCCc2c(O)[nH]c3nc(N)nc(N)c23)cc1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DHFR P00374 6/20 0.37
CYP4A11 Q02928 2/20 0.35
NAMPT P43490 2/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
CA14 Q9ULX7 1/20 0.35
TYMS P04818 1/20 0.35
DHODH Q02127 1/20 0.35
TLR8 Q9NR97 1/20 0.35
TLR7 Q9NYK1 1/20 0.35
CYP4F2 P78329 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8997191 0.83 DHFR (0.36) DHFRCA12CA1CA2CA9
SCHEMBL9859911 0.82 FOLR1 (0.36) DHFR
SCHEMBL8997147 0.81 NAMPT (0.50) DHFRNAMPTTYMS
SCHEMBL9042476 0.77 LMNA (0.34) DHFRCA12CA1CA2CA9
SCHEMBL8997169 0.75 DHFR (0.50) DHFRTYMS
SCHEMBL8997185 0.75 DHFR (0.50) DHFRTYMS
SCHEMBL9039740 0.74 DHFR (0.51) DHFR
SCHEMBL9446114 0.74 DHFR (0.46) DHFR
SCHEMBL8997157 0.74 DHFR (0.65) DHFRTYMS
SCHEMBL9042926 0.73 DHFR (0.41) DHFRNAMPTTYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0334636-B1 Pyrrolopyrimidine derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1996-10-23 EP disclosed
US-5539113-A ANTITUMOR AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-07-23 US disclosed
US-5296600-A Antitumor agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-03-22 US disclosed
US-5106974-A Antitumor and -carcinogenic agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-04-21 US disclosed
US-4997838-A Antitumor agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1991-03-05 US disclosed
EP-0334636-A2 Pyrrolopyrimidine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1989-09-27 EP disclosed