SCHEMBL8997157

SCHEMBL8997157

Nc1nc(N)c2c(CCCc3ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc3)c(O)[nH]c2n1

nearest known ligand 0.65

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DHFR P00374 11/20 0.65
GART P22102 3/20 0.64
ATIC P31939 1/20 0.64
TYMS P04818 4/20 0.63
FOLR2 P14207 1/20 0.56
FOLR1 P15328 1/20 0.56
SLC19A1 P41440 1/20 0.56
SLC46A1 Q96NT5 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9085889 0.91 DHFR (0.75) DHFRGARTATICTYMSFOLR2
SCHEMBL9087509 0.89 DHFR (0.67) DHFRGARTATICTYMSFOLR2
SCHEMBL9088158 0.88 DHFR (0.61) DHFRGARTATICTYMSFOLR2
SCHEMBL9088410 0.88 GART (0.62) DHFRGARTATICTYMSFOLR2
SCHEMBL9343717 0.87 DHFR (0.74) DHFRGARTATICTYMSFOLR2
SCHEMBL9339203 0.85 DHFR (0.69) DHFRGARTATICTYMSFOLR2
SCHEMBL9339239 0.85 GART (0.75) DHFRGARTATICTYMSFOLR2
SCHEMBL8997169 0.84 DHFR (0.50) DHFRGARTATICTYMS
SCHEMBL8997185 0.84 DHFR (0.50) DHFRGARTATICTYMS
SCHEMBL9339217 0.84 GART (0.74) DHFRGARTATICTYMSFOLR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4997838-A Antitumor agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1991-03-05 US claimed
EP-0334636-B1 Pyrrolopyrimidine derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1996-10-23 EP disclosed
US-5539113-A ANTITUMOR AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-07-23 US disclosed
US-5296600-A Antitumor agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-03-22 US disclosed
US-5106974-A Antitumor and -carcinogenic agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-04-21 US disclosed
US-4997838-A Antitumor agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1991-03-05 US disclosed
EP-0334636-A2 Pyrrolopyrimidine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1989-09-27 EP disclosed