SCHEMBL8997164

SCHEMBL8997164

CCOC(=O)CC[C@@H](NC(=O)c1ccc(CCCC2CNc3nc(N)nc(O)c32)cc1)C(=O)OCC

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DHFR P00374 3/20 0.44
GART P22102 4/20 0.44
ATIC P31939 2/20 0.44
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
HSD17B10 Q99714 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8997156 1.00 DHFR (0.44) DHFRGARTATICKDM4EALDH1A1
SCHEMBL8997167 0.95 ATIC (0.47) DHFRGARTATICKDM4EALDH1A1
SCHEMBL8997175 0.95 ATIC (0.47) DHFRGARTATICKDM4EALDH1A1
SCHEMBL8997230 0.93 DHFR (0.50) DHFRGARTATICKDM4EALDH1A1
SCHEMBL8997237 0.93 DHFR (0.50) DHFRGARTATICKDM4EALDH1A1
SCHEMBL9446079 0.87 GART (0.51) DHFRGARTATICKDM4EALDH1A1
SCHEMBL9446085 0.87 GART (0.51) DHFRGARTATICKDM4EALDH1A1
SCHEMBL9859650 0.87 GART (0.42) DHFRGARTATICKDM4EALDH1A1
SCHEMBL9859644 0.87 GART (0.42) DHFRGARTATICKDM4EALDH1A1
SCHEMBL9844816 0.85 DHFR (0.42) DHFRGARTKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4997838-A Antitumor agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1991-03-05 US claimed
EP-0334636-B1 Pyrrolopyrimidine derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1996-10-23 EP disclosed
US-5539113-A ANTITUMOR AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-07-23 US disclosed
US-5106974-A Antitumor and -carcinogenic agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-04-21 US disclosed
US-4997838-A Antitumor agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1991-03-05 US disclosed
EP-0334636-A2 Pyrrolopyrimidine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1989-09-27 EP disclosed