SCHEMBL9859650

SCHEMBL9859650

CCOC(=O)CC[C@@H](NC(=O)c1ccc(CCCC2CNc3nc(N)nc(O)c32)s1)C(=O)OCC

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GART P22102 7/20 0.42
DHFR P00374 3/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
FOLR1 P15328 9/20 0.38
SLC46A1 Q96NT5 7/20 0.38
SLC19A1 P41440 4/20 0.38
FOLR2 P14207 3/20 0.37
ATIC P31939 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9859644 1.00 GART (0.42) GARTDHFRKDM4EALDH1A1HPGD
SCHEMBL9439735 0.93 DHFR (0.43) GARTDHFRKDM4EALDH1A1HPGD
SCHEMBL9439730 0.93 DHFR (0.43) GARTDHFRKDM4EALDH1A1HPGD
SCHEMBL8997156 0.87 DHFR (0.44) GARTDHFRKDM4EALDH1A1HPGD
SCHEMBL8997164 0.87 DHFR (0.44) GARTDHFRKDM4EALDH1A1HPGD
SCHEMBL9439358 0.85 GART (0.58) GARTFOLR1SLC46A1SLC19A1FOLR2
SCHEMBL8997175 0.83 ATIC (0.47) GARTDHFRKDM4EALDH1A1HPGD
SCHEMBL8997167 0.83 ATIC (0.47) GARTDHFRKDM4EALDH1A1HPGD
SCHEMBL9439621 0.80 DHFR (0.40) GARTDHFRALDH1A1HPGDL3MBTL1
SCHEMBL8997230 0.80 DHFR (0.50) GARTDHFRKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0418924-A2 Pyrrolopyrimidines, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-03-27 EP disclosed