SCHEMBL8997262

SCHEMBL8997262

Cn1ncc(C#N)c1N(C(=O)c1ccc(Cl)cc1)C(N)=S

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
ALDH1A1 P00352 4/20 0.35
NPC1 O15118 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
HTT P42858 1/20 0.35
XDH P47989 1/20 0.34
KMT2A Q03164 3/20 0.34
F2 P00734 1/20 0.34
MAP4K4 O95819 2/20 0.33
MEN1 O00255 2/20 0.33
HPGD P15428 2/20 0.33
KDM4E B2RXH2 2/20 0.33
LMNA P02545 2/20 0.33
POLB P06746 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
ITK Q08881 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20540301 0.72 MAPT (0.45) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL8997249 0.69 CYP1A2 (0.56) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL8997267 0.68 CYP3A4 (0.51) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL8997211 0.67 MAPT (0.40) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL6326170 0.65 POLB (0.37) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL6174901 0.63 POLB (0.41) CYP1A2CYP2C19ALDH1A1L3MBTL1HTT
SCHEMBL27706292 0.62 CES2 (0.46) CYP3A4CYP2C19ALDH1A1NPC1L3MBTL1
SCHEMBL28601701 0.61 MEN1 (0.49) ALDH1A1NPC1HTTKMT2AMEN1
SCHEMBL11090784 0.60 LMNA (0.42) ALDH1A1L3MBTL1KMT2AMEN1KDM4E
SCHEMBL4520111 0.60

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5486618-A PLANT SAFENING AGENTS BASF AKTIENGESELLSCHAFT (DE) 1996-01-23 US disclosed
EP-0561836-A1 SUBSTITUTED 5-AMINOPYRAZOLS BASF Aktiengesellschaft (DE) 1993-09-29 EP disclosed
WO-1992010480-A1 SUBSTITUTED 5-AMINOPYRAZOLS BASF AKTIENGESELLSCHAFT (DE) 1992-06-25 WO disclosed