SCHEMBL8997570

SCHEMBL8997570

COc1cccc2c1C[C@@](NC(=O)c1ccccc1)(C(=O)c1[c]cccc1)CC2

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 2/20 0.46
MTNR1B P49286 2/20 0.46
CXCR5 P32302 2/20 0.38
HDAC1 Q13547 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
ADRA2A P08913 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
HCN1 O60741 1/20 0.35
HCN4 Q9Y3Q4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8583793 0.85 MTNR1A (0.54) MTNR1AMTNR1BCXCR5HDAC1HDAC6
SCHEMBL8583790 0.85 MTNR1A (0.54) MTNR1AMTNR1BCXCR5HDAC1HDAC6
SCHEMBL8584280 0.85 MTNR1A (0.54) MTNR1AMTNR1BCXCR5HDAC1HDAC6
SCHEMBL8599195 0.74 MTNR1A (0.51) MTNR1AMTNR1BHDAC1HDAC6ADRA2A
SCHEMBL8598490 0.74 MTNR1A (0.51) MTNR1AMTNR1BHDAC1HDAC6ADRA2A
SCHEMBL8845587 0.71 MTNR1A (0.45) MTNR1AMTNR1BCXCR5ADRA2ANPC1
SCHEMBL8596061 0.70 MMP1 (0.48) MTNR1AMTNR1B
SCHEMBL8424174 0.70 CXCR5 (0.50) CXCR5
SCHEMBL8424334 0.70 CXCR5 (0.50) CXCR5
SCHEMBL8422478 0.70 CXCR5 (0.50) CXCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729972-A1 Peptide derivatives of tetrahydronaphthalene F. HOFFMANN-LA ROCHE AG (CH) 1996-09-04 EP disclosed