SCHEMBL8998740

SCHEMBL8998740

CCc1ncoc1C(N)=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GLA P06280 1/20 0.37
ADORA2A P29274 1/20 0.35
GABRP O00591 1/20 0.33
GABRD O14764 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRB1 P18505 1/20 0.33
GABRG2 P18507 1/20 0.33
GABRB3 P28472 1/20 0.33
GABRA5 P31644 1/20 0.33
GABRA3 P34903 1/20 0.33
GABRA2 P47869 1/20 0.33
GABRB2 P47870 1/20 0.33
GABRA4 P48169 1/20 0.33
GABRE P78334 1/20 0.33
GABRA6 Q16445 1/20 0.33
GABRG1 Q8N1C3 1/20 0.33
GABRG3 Q99928 1/20 0.33
GABRQ Q9UN88 1/20 0.33
KMT2A Q03164 4/20 0.32
MEN1 O00255 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17826659 0.82 KMT2A (0.33) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL2570641 0.82 KMT2A (0.40) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL29290254 0.81 GLA (0.37) GLAADORA2AKMT2AMEN1ALDH1A1
SCHEMBL22018447 0.78 GLA (0.36) GLAADORA2AKMT2ALMNA
SCHEMBL8518849 0.77 ADORA2A (0.33) GLAADORA2A
SCHEMBL2139234 0.74
SCHEMBL11879772 0.71 ADORA2A (0.52) GLAADORA2AKMT2AMEN1NPC1
SCHEMBL2592947 0.69 ADORA2A (0.46) GLAADORA2ANPC1RAB9APARP10
SCHEMBL14311731 0.69
SCHEMBL9004531 0.66

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0492233-B1 Method for the preparation of 5-cyano-4-alkyl-oxazol HOFFMANN LA ROCHE (CH) 1996-08-21 EP claimed
EP-0492233-A1 Method for the preparation of 5-cyano-4-alkyl-oxazol F. HOFFMANN-LA ROCHE AG (CH) 1992-07-01 EP claimed
EP-4630115-A1 THERAPEUTIC COMPOUNDS Sanofi (FR) 2025-10-15 EP disclosed
WO-2025104230-A1 BENZOXAZOLES AS MODULATORS OF IL-17A SANOFI (FR) 2025-05-22 WO disclosed
WO-2024121427-A1 THERAPEUTIC COMPOUNDS SANOFI (FR) 2024-06-13 WO disclosed
US-11939343-B2 Sting agonist compounds and methods of use MERSANA THERAPEUTICS, INC. (US) 2024-03-26 US disclosed
CN-114585623-A Bis [ N- ((5-carbamoyl) -1H-benzo [ d ] imidazol-2-yl) pyrazole-5-carboxamide ] derivatives and related compounds as STING (interferon gene stimulator) agonists for the treatment of cancer 梅尔莎纳医疗公司 2022-06-03 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11939343-B2 Sting agonist compounds and methods of use STING1, IRF3, MAVS GLA 2351/4885ADORA2A 267/4885GABRP 808/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.