SCHEMBL8998884

SCHEMBL8998884

Cn1c(Br)c(C=O)c2ccccc21

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.60
LMNA P02545 2/20 0.60
CYP1A2 P05177 2/20 0.59
CYP2C19 P33261 2/20 0.59
POLB P06746 2/20 0.59
HTT P42858 7/20 0.57
NPSR1 Q6W5P4 6/20 0.57
MAPT P10636 5/20 0.57
SMN1; SMN2 Q16637 3/20 0.57
HPGD P15428 2/20 0.55
CYP3A4 P08684 1/20 0.55
L3MBTL1 Q9Y468 2/20 0.54
ATM Q13315 1/20 0.50
NOD2 Q9HC29 1/20 0.50
GPR3 P46089 1/20 0.48
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
IMPDH2 P12268 1/20 0.44
AHR P35869 1/20 0.44
KDM4E B2RXH2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1792194 0.79 ALDH1A1 (0.62) ALDH1A1LMNACYP1A2CYP2C19POLB
SCHEMBL30534146 0.79 ALDH1A1 (0.62) ALDH1A1LMNACYP1A2CYP2C19POLB
SCHEMBL26631812 0.78 ALDH1A1 (0.60) ALDH1A1LMNACYP1A2CYP2C19POLB
SCHEMBL14519065 0.78 ALDH1A1 (0.60) ALDH1A1LMNACYP1A2CYP2C19POLB
SCHEMBL1092518 0.78 ALDH1A1 (0.60) ALDH1A1LMNACYP1A2CYP2C19POLB
SCHEMBL29374992 0.78 ALDH1A1 (0.60) ALDH1A1LMNACYP1A2CYP2C19POLB
SCHEMBL671977 0.77 POLB (0.44) ALDH1A1LMNACYP1A2CYP2C19POLB
SCHEMBL22443301 0.75 L3MBTL1 (0.52) ALDH1A1LMNACYP1A2CYP2C19POLB
SCHEMBL1429358 0.75 ALDH1A1 (1.00) ALDH1A1LMNACYP1A2CYP2C19POLB
SCHEMBL25708943 0.75 POLB (0.48) ALDH1A1LMNACYP1A2CYP2C19POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109912576-A Cyclic annular or loop coil Diamines pyrimidine-hydroxamic acid and application thereof 华东理工大学 2019-06-21 CN disclosed
CN-104610355-B Indole framework based center chirality sulfonamides monophosphine ligand and preparation method 华东师范大学 2017-01-11 CN disclosed
US-5556874-A ENZYME INHIBITORS AS ANTICARCINOGENIC AGENTS WARNER LAMBERT COMPANY (US) 1996-09-17 US disclosed
US-5464861-A Anticarcinogenic agents WARNER-LAMBERT (US) 1995-11-07 US disclosed
EP-0654024-A1 2-THIOINDOLES (SELENOINDOLES) AND RELATED DISULFIDES (SELENIDES) WHICH INHIBIT PROTEIN TYROSINE KINASES AND WHICH HAVE ANTITUMOR PROPERTIES WARNER-LAMBERT COMPANY (US) 1995-05-24 EP disclosed
WO-1994003427-A1 2-THIOINDOLES (SELENOINDOLES) AND RELATED DISULFIDES (SELENIDES) WHICH INHIBIT PROTEIN TYROSINE KINASES AND WHICH HAVE ANTITUMOR PROPERTIES WARNER-LAMBERT COMPANY (US) 1994-02-17 WO disclosed