SCHEMBL8998915

SCHEMBL8998915

Cn1c(SSc2c(C(=O)Nc3ccncc3)c3ccccc3n2C)c(C(=O)Nc2ccncc2)c2ccccc21

nearest known ligand 0.81

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SRC P12931 18/20 0.81
EGFR P00533 14/20 0.81
FGFR1 P11362 1/20 0.81
NPC1 O15118 1/20 0.59
ALDH1A1 P00352 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1527703 0.89 SRC (1.00) SRCEGFRFGFR1NPC1ALDH1A1
SCHEMBL8999317 0.86 SRC (0.75) SRCEGFRFGFR1NPC1ALDH1A1
SCHEMBL8999141 0.86 NPC1 (0.80) SRCEGFRFGFR1NPC1ALDH1A1
SCHEMBL8998829 0.84 SRC (1.00) SRCEGFRFGFR1NPC1ALDH1A1
SCHEMBL8999420 0.81 SRC (1.00) SRCEGFRFGFR1
SCHEMBL8998908 0.81 SRC (1.00) SRCEGFRFGFR1NPC1ALDH1A1
SCHEMBL8999355 0.79 SRC (0.67) SRCEGFRFGFR1
SCHEMBL15708776 0.79 ALDH1A1 (0.54) SRCEGFRFGFR1NPC1ALDH1A1
SCHEMBL30919366 0.79 ALDH1A1 (0.54) SRCEGFRFGFR1NPC1ALDH1A1
SCHEMBL8999067 0.78 SRC (1.00) SRCEGFRFGFR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5556874-A ENZYME INHIBITORS AS ANTICARCINOGENIC AGENTS WARNER LAMBERT COMPANY (US) 1996-09-17 US disclosed
US-5464861-A Anticarcinogenic agents WARNER-LAMBERT (US) 1995-11-07 US disclosed
EP-0654024-A1 2-THIOINDOLES (SELENOINDOLES) AND RELATED DISULFIDES (SELENIDES) WHICH INHIBIT PROTEIN TYROSINE KINASES AND WHICH HAVE ANTITUMOR PROPERTIES WARNER-LAMBERT COMPANY (US) 1995-05-24 EP disclosed
WO-1994003427-A1 2-THIOINDOLES (SELENOINDOLES) AND RELATED DISULFIDES (SELENIDES) WHICH INHIBIT PROTEIN TYROSINE KINASES AND WHICH HAVE ANTITUMOR PROPERTIES WARNER-LAMBERT COMPANY (US) 1994-02-17 WO disclosed