SCHEMBL9000486

SCHEMBL9000486

C(=Cc1nc(C=Cc2cncc(-c3cccc4ccccc34)c2)c(C=Cc2cncc(-c3cccc4ccccc34)c2)nc1C=Cc1cncc(-c2cccc3ccccc23)c1)c1cncc(-c2cccc3ccccc23)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
CHRNB1 P11230 1/20 0.41
CHRNB2 P17787 1/20 0.41
CHRNB4 P30926 1/20 0.41
CHRNA3 P32297 1/20 0.41
CHRNB3 Q05901 1/20 0.41
TNF P01375 1/20 0.40
KDM4E B2RXH2 3/20 0.38
ALDH1A1 P00352 3/20 0.38
MAPT P10636 3/20 0.38
HPGD P15428 3/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
RAB9A P51151 2/20 0.38
CA12 O43570 1/20 0.38
CA9 Q16790 1/20 0.38
AKT1 P31749 3/20 0.37
CYP11B1 P15538 2/20 0.36
CYP11B2 P19099 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9000337 0.78 CYP11B1 (0.44) KDM1AHDAC1HDAC6ALDH1A1RAB9A
SCHEMBL9000353 0.76 CYP11B2 (0.50) CHRNB1CHRNB2CHRNB4CHRNA3CHRNB3
SCHEMBL30963861 0.73 CYP11B1 (0.53) HDAC6CHRNB1CHRNB2CHRNB4CHRNA3
SCHEMBL30963859 0.73 CYP11B1 (0.53) HDAC6CHRNB1CHRNB2CHRNB4CHRNA3
SCHEMBL16805019 0.73 CHRNB1 (0.45) CHRNB1CHRNB2CHRNB4CHRNA3CHRNB3
SCHEMBL9000571 0.73 HDAC8 (0.41) HDAC6CHRNB4CHRNA3TNFKDM4E
SCHEMBL9000391 0.72 CYP11B1 (0.46) KDM4EALDH1A1MAPTHPGDSMN1; SMN2
SCHEMBL9000334 0.71 CA12 (0.38) TNFKDM4EALDH1A1MAPTHPGD
SCHEMBL9000346 0.71 KDM1A (0.47) KDM1AHDAC1HDAC6KDM4EALDH1A1
SCHEMBL18253148 0.70 TNF (0.52) HDAC6TNFKDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0516409-B1 Tetravinylpyrazine compound, method for preparing same and electroluminescent element and non-linear optical material using same MITSUI TOATSU CHEMICALS (JP) 1996-09-11 EP disclosed
US-5416213-A Tetravinylpyrazine compound, method for preparing same and electroluminescent element and non-linear optical material using same MITSUI TOATSU CHEMICALS, INC. (JP) 1995-05-16 US disclosed
EP-0516409-A2 Tetravinylpyrazine compound, method for preparing same and electroluminescent element and non-linear optical material using same MITSUI TOATSU CHEMICALS, Inc. (JP) 1992-12-02 EP disclosed