SCHEMBL9001822

SCHEMBL9001822

CC(CC1CCc2nc(N)nc(O)c21)c1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)s1

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DHFR P00374 3/20 0.43
MTR Q99707 1/20 0.43
GART P22102 4/20 0.39
FOLR1 P15328 5/20 0.38
ATIC P31939 3/20 0.38
FOLR2 P14207 2/20 0.37
SLC19A1 P41440 1/20 0.37
SLC46A1 Q96NT5 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8567075 0.93 DHFR (0.47) DHFRMTRGART
SCHEMBL9001764 0.90 DHFR (0.42) DHFRMTRGART
SCHEMBL9001907 0.86 DHFR (0.53) DHFRMTRATIC
SCHEMBL8566521 0.85 DHFR (0.46) DHFRMTRGART
SCHEMBL9001752 0.83 GART (0.53) GARTFOLR1ATICFOLR2SLC19A1
SCHEMBL9001769 0.82 FOLR1 (0.49) GARTFOLR1ATICFOLR2SLC19A1
SCHEMBL9001765 0.79 DHFR (0.52) DHFRMTRATIC
SCHEMBL8570088 0.78 DHFR (0.58) DHFRMTR
SCHEMBL9001801 0.76 DHFR (0.53) DHFRMTRGARTATIC
SCHEMBL9001799 0.75 DHFR (0.54) DHFRMTRGARTATIC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed