SCHEMBL9001799

SCHEMBL9001799

Nc1nc(O)c2c(n1)CCC2CCCc1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc1

nearest known ligand 0.86

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DHFR P00374 8/20 0.54
GART P22102 3/20 0.53
MTR Q99707 1/20 0.51
ATIC P31939 1/20 0.50
TYMS P04818 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9001801 0.95 DHFR (0.53) DHFRGARTMTRATICTYMS
SCHEMBL1066004 0.92 DHFR (0.59) DHFRGARTMTRATIC
SCHEMBL9001930 0.88 ATIC (0.48) DHFRGARTMTRATICTYMS
SCHEMBL8571475 0.87 DHFR (0.57) DHFRGARTMTR
SCHEMBL9001769 0.85 FOLR1 (0.49) GARTATIC
SCHEMBL9446088 0.85 GART (0.53) DHFRGARTMTRATIC
SCHEMBL8997205 0.85 GART (0.60) DHFRGARTATICTYMS
SCHEMBL9001791 0.84 ATIC (0.46) DHFRGARTMTRATICTYMS
SCHEMBL9001907 0.84 DHFR (0.53) DHFRMTRATIC
SCHEMBL9844814 0.83 DHFR (0.52) DHFRGARTATICTYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP claimed
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP disclosed