SCHEMBL8567075

SCHEMBL8567075

CC(CC1CCc2nc(N)nc(N)c21)c1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)s1

nearest known ligand 0.61

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DHFR P00374 6/20 0.47
MTR Q99707 3/20 0.47
GART P22102 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8566521 0.93 DHFR (0.46) DHFRMTRGART
SCHEMBL9001822 0.93 DHFR (0.43) DHFRMTRGART
SCHEMBL8570088 0.85 DHFR (0.58) DHFRMTR
SCHEMBL9001764 0.83 DHFR (0.42) DHFRMTRGART
SCHEMBL8563180 0.82 FOLR1 (0.51) DHFRMTRGART
SCHEMBL9439711 0.79 GART (0.49) DHFRGART
SCHEMBL8569142 0.78 DHFR (0.59) DHFRMTR
SCHEMBL9001907 0.78 DHFR (0.53) DHFRMTR
SCHEMBL8571475 0.76 DHFR (0.57) DHFRMTRGART
SCHEMBL9001752 0.76 GART (0.53) GART

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530579-B1 Condensed pyrimidine derivatives antitumor agents EISAI CO LTD (JP) 1998-11-11 EP disclosed
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed