SCHEMBL9002415

SCHEMBL9002415

O=S(=O)(NCCCOc1cccc2nccn12)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.51
F13A1 P00488 3/20 0.51
ALDH1A1 P00352 6/20 0.48
TSHR P16473 1/20 0.48
KDM4E B2RXH2 1/20 0.48
LMNA P02545 1/20 0.48
PKM P14618 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
GLRA3 O75311 1/20 0.47
GLRB P48167 1/20 0.47
CDK2 P24941 2/20 0.44
CDK1 P06493 1/20 0.44
CDK4 P11802 1/20 0.44
MAPT P10636 1/20 0.42
TDP1 Q9NUW8 1/20 0.41
TBXA2R P21731 1/20 0.41
MEN1 O00255 1/20 0.41
HTT P42858 1/20 0.41
KMT2A Q03164 1/20 0.41
BRAF P15056 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9001991 0.84 POLB (0.38) F13A1ALDH1A1KDM4EPKMCDK2
SCHEMBL9002369 0.83 CYP3A4 (0.50) ALDH1A1KDM4ELMNASMN1; SMN2MEN1
SCHEMBL9001957 0.81 IDO1 (0.43) F13A1CDK2CDK1CDK4MEN1
SCHEMBL9002403 0.81 CYP4F2 (0.41) F13A1ALDH1A1CDK2CDK1CDK4
SCHEMBL9002512 0.80 HTT (0.41) ALDH1A1KDM4EPKMCDK2CDK1
SCHEMBL9002438 0.80 CYP3A4 (0.46) ALDH1A1KDM4ELMNASMN1; SMN2GLRA3
SCHEMBL9001970 0.80 CYP4F2 (0.42) F13A1ALDH1A1CDK2CDK1CDK4
SCHEMBL9002264 0.80 CYP4F2 (0.42) F13A1ALDH1A1CDK2CDK1CDK4
SCHEMBL9002497 0.79 ALDH1A1 (0.54) MAPK1F13A1ALDH1A1TSHRKDM4E
SCHEMBL9001987 0.78 GLO1 (0.41) ALDH1A1KDM4ESMN1; SMN2GLRA3GLRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5587383-A CALMODULIN INHIBITORS; ANTIISCHEMIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-12-24 US disclosed
EP-0471236-B1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-03-15 EP disclosed
US-5395839-A Calmodulin and angiogenesis inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-03-07 US disclosed
US-5244908-A Calmodulin inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-09-14 US disclosed
EP-0471236-A1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-02-19 EP disclosed