SCHEMBL9002019

SCHEMBL9002019

CS(=O)(=O)NCCOCCSc1cccc2nccn12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.35
MAPT P10636 2/20 0.35
MEN1 O00255 1/20 0.34
HTT P42858 1/20 0.34
KMT2A Q03164 1/20 0.34
HSD17B10 Q99714 1/20 0.33
RECQL P46063 1/20 0.33
ROCK1 Q13464 3/20 0.32
CDK8 P49336 2/20 0.32
CLK4 Q9HAZ1 2/20 0.32
FLT1 P17948 1/20 0.32
CDK9 P50750 1/20 0.32
LIMK1 P53667 1/20 0.32
MAP4K4 O95819 2/20 0.32
PRKACA P17612 2/20 0.32
MAP4K2 Q12851 2/20 0.32
DYRK1A Q13627 2/20 0.32
AURKB Q96GD4 2/20 0.32
KCNJ5 P48544 1/20 0.32
KCNJ3 P48549 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9002172 0.88 MAPT (0.43) ALDH1A1MAPTMEN1HTTKMT2A
Hydrochloric Acid SCHEMBL9001908 0.87 MAPT (0.42) ALDH1A1MAPTMEN1HTTKMT2A
SCHEMBL9002013 0.86 POLB (0.37) ALDH1A1MAPTHTTHSD17B10RECQL
SCHEMBL9002010 0.85 POLB (0.36) ALDH1A1MAPTMEN1HTTKMT2A
SCHEMBL9001996 0.81 CDK8 (0.35) ROCK1CDK8CLK4FLT1CDK9
SCHEMBL9002027 0.78 CNR2 (0.36) ALDH1A1MAPTMEN1HTTKMT2A
SCHEMBL9002512 0.77 HTT (0.41) ALDH1A1MAPTMEN1HTTKMT2A
SCHEMBL9002373 0.77 KDM4E (0.36) ALDH1A1MAPTMEN1KMT2AHSD17B10
SCHEMBL9002414 0.77 CDK8 (0.34) ALDH1A1MAPTMEN1HTTKMT2A
SCHEMBL9002262 0.76 NPY5R (0.33) ALDH1A1MAPTMEN1HTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5587383-A CALMODULIN INHIBITORS; ANTIISCHEMIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-12-24 US disclosed
EP-0471236-B1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-03-15 EP disclosed
US-5395839-A Calmodulin and angiogenesis inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-03-07 US disclosed
US-5244908-A Calmodulin inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-09-14 US disclosed
EP-0471236-A1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-02-19 EP disclosed