SCHEMBL9001996

SCHEMBL9001996

CS(=O)(=O)OCCSc1cccc2nccn12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK8 P49336 2/20 0.35
ROCK1 Q13464 2/20 0.35
CHEK1 O14757 2/20 0.35
MAP4K4 O95819 1/20 0.35
CSF1R P07333 1/20 0.35
PRKACA P17612 1/20 0.35
KDR P35968 1/20 0.35
MAP2K1 Q02750 1/20 0.35
ACVR1 Q04771 1/20 0.35
MAP4K2 Q12851 1/20 0.35
DYRK1A Q13627 1/20 0.35
AURKB Q96GD4 1/20 0.35
DYRK1B Q9Y463 1/20 0.35
FLT1 P17948 1/20 0.35
CDK9 P50750 1/20 0.35
LIMK1 P53667 1/20 0.35
CLK4 Q9HAZ1 1/20 0.35
ADORA3 P0DMS8 1/20 0.31
ATR Q13535 1/20 0.30
PDCD1 Q15116 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9002414 0.93 CDK8 (0.34) CDK8ROCK1CHEK1MAP4K4CSF1R
SCHEMBL7846687 0.88 CDK8 (0.32) CDK8ROCK1CHEK1MAP4K4CSF1R
SCHEMBL9002019 0.81 ALDH1A1 (0.35) CDK8ROCK1CHEK1MAP4K4CSF1R
SCHEMBL8581462 0.80 PTGS2 (0.36) CDK8ROCK1CHEK1MAP4K4CSF1R
SCHEMBL9002172 0.80 MAPT (0.43) CDK8ROCK1CHEK1MAP4K4CSF1R
Hydrochloric Acid SCHEMBL9001908 0.79 MAPT (0.42) CDK8ROCK1CHEK1MAP4K4CSF1R
SCHEMBL9002463 0.79 CDK8 (0.35) CDK8ROCK1CHEK1MAP4K4CSF1R
Hydrochloric Acid SCHEMBL9185489 0.78 CDK8 (0.34) CDK8ROCK1CHEK1MAP4K4CSF1R
SCHEMBL9002013 0.78 POLB (0.37) CDK8ROCK1CHEK1MAP4K4CSF1R
SCHEMBL9001943 0.77 CDK8 (0.38) CDK8ROCK1CHEK1MAP4K4CSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5587383-A CALMODULIN INHIBITORS; ANTIISCHEMIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-12-24 US disclosed
EP-0471236-B1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-03-15 EP disclosed
US-5395839-A Calmodulin and angiogenesis inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-03-07 US disclosed
US-5244908-A Calmodulin inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-09-14 US disclosed
EP-0471236-A1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-02-19 EP disclosed