SCHEMBL9002373

SCHEMBL9002373

CCCS(=O)(=O)NCCSc1cccc2nccn12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.36
HSD17B10 Q99714 1/20 0.36
TP53 P04637 5/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
HTR6 P50406 1/20 0.33
NPC1 O15118 2/20 0.33
TSHR P16473 1/20 0.33
RAB9A P51151 1/20 0.33
CDK8 P49336 2/20 0.33
ROCK1 Q13464 2/20 0.33
FLT1 P17948 1/20 0.33
CDK9 P50750 1/20 0.33
LIMK1 P53667 1/20 0.33
CLK4 Q9HAZ1 1/20 0.33
CHEK1 O14757 1/20 0.33
MAP4K4 O95819 1/20 0.33
CSF1R P07333 1/20 0.33
PRKACA P17612 1/20 0.33
KDR P35968 1/20 0.33
MAP2K1 Q02750 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9002291 0.93 HPGD (0.35) KDM4EHSD17B10CDK8ROCK1FLT1
SCHEMBL9002027 0.92 CNR2 (0.36) KDM4EHSD17B10SMN1; SMN2TSHRRAB9A
SCHEMBL9001931 0.91 KDM4E (0.39) KDM4EMAPTALDH1A1GAA
SCHEMBL9002012 0.91 KDM4E (0.39) KDM4EMAPTALDH1A1GAA
SCHEMBL9002202 0.87 CHEK1 (0.32) CDK8ROCK1CHEK1MAP4K4CSF1R
SCHEMBL9002172 0.85 MAPT (0.43) HSD17B10TSHRCDK8ROCK1FLT1
Hydrochloric Acid SCHEMBL9001908 0.84 MAPT (0.42) HSD17B10TSHRCDK8ROCK1FLT1
SCHEMBL9002262 0.82 NPY5R (0.33) HSD17B10TSHRCDK8ROCK1FLT1
SCHEMBL9001975 0.80 KMT2A (0.47) KDM4EHSD17B10TP53SMN1; SMN2TSHR
SCHEMBL9002538 0.80 CDK8 (0.33) CDK8ROCK1FLT1CDK9LIMK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5587383-A CALMODULIN INHIBITORS; ANTIISCHEMIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-12-24 US disclosed
EP-0471236-B1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-03-15 EP disclosed
US-5395839-A Calmodulin and angiogenesis inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-03-07 US disclosed
US-5244908-A Calmodulin inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-09-14 US disclosed
EP-0471236-A1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-02-19 EP disclosed